SCHEMBL29640863

SCHEMBL29640863

C(#Cn1ncc2ccccc21)c1ccnc(-c2ccnc(N3CCN(c4ncc[nH]4)CC3)n2)n1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 14/20 0.37
DKK1 O94907 2/20 0.32
CCNT1 O60563 2/20 0.31
CCNA2 P20248 2/20 0.31
CDK2 P24941 2/20 0.31
CDK9 P50750 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640843 0.86 MAPT (0.40) DYRK1A
SCHEMBL29640876 0.83 DYRK1A (0.37) DYRK1A
SCHEMBL29640867 0.83 CYP11B2 (0.38) DYRK1A
SCHEMBL29640810 0.82 DYRK1A (0.36) DYRK1A
SCHEMBL29640870 0.81 ACACB (0.43) DYRK1ADKK1
SCHEMBL29640903 0.78 DYRK1A (0.38) DYRK1ADKK1CDK2
SCHEMBL29640982 0.78 ROCK2 (0.42) DYRK1A
SCHEMBL29640839 0.77 DYRK1A (0.34) DYRK1A
SCHEMBL29640778 0.76 ROCK2 (0.38) DYRK1A
SCHEMBL29640817 0.76 DYRK1A (0.37) DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed