SCHEMBL29640899

SCHEMBL29640899

Brc1ccnc(-c2ccncn2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LATS1 O95835 3/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HSP90AA1 P07900 1/20 0.34
MAPK9 P45984 3/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPK13 O15264 1/20 0.34
RAF1 P04049 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34
ADORA2A P29274 2/20 0.33
ADORA2B P29275 2/20 0.33
ADORA1 P30542 2/20 0.33
NPC1 O15118 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAP4K4 O95819 2/20 0.32
EGFR P00533 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640832 0.77 MAPK9 (0.37) LATS1MEN1KMT2AHSP90AA1MAPK9
SCHEMBL29640833 0.77 MAPK9 (0.37) LATS1MEN1KMT2AHSP90AA1MAPK9
SCHEMBL38655465 0.75 GRM5 (0.46) MEN1KMT2AMAPK9ALDH1A1MAPK13
SCHEMBL29627704 0.74 HSP90AA1 (0.42) LATS1HSP90AA1MAPK9KDM4EALDH1A1
SCHEMBL6449580 0.74 HSP90AA1 (0.42) LATS1HSP90AA1MAPK9KDM4EALDH1A1
SCHEMBL8891318 0.74 KDM4E (0.65) HSP90AA1KDM4EALDH1A1NPC1TDP1
SCHEMBL2679072 0.74 NPC1 (0.47) MEN1KMT2ANPC1MAPT
SCHEMBL8892702 0.73 NPC1 (0.44) KDM4EADORA2AADORA1NPC1TDP1
SCHEMBL25295479 0.72 TP53 (0.48) LATS1HSP90AA1MAPK9MAPK13RAF1
SCHEMBL5989213 0.72 HSP90AA1 (0.44) LATS1HSP90AA1MAPK9MAPK13RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed