SCHEMBL29640833

SCHEMBL29640833

Clc1ccnc(-c2ccncn2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK9 P45984 3/20 0.37
MAP4K4 O95819 3/20 0.37
EGFR P00533 2/20 0.37
FRK P42685 2/20 0.37
CSNK1A1 P48729 2/20 0.37
DCLK1 O15075 1/20 0.37
PRKD3 O94806 1/20 0.37
PRKACA P17612 1/20 0.37
FLT3 P36888 1/20 0.37
GSK3B P49841 1/20 0.37
MINK1 Q8N4C8 1/20 0.37
SLK Q9H2G2 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
MAP4K5 Q9Y4K4 1/20 0.37
MAPK14 Q16539 2/20 0.36
RPS6KA5 O75582 1/20 0.36
RPS6KA4 O75676 1/20 0.36
MAPK10 P53779 1/20 0.36
MAPT P10636 3/20 0.35
MEN1 O00255 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640832 1.00 MAPK9 (0.37) MAPK9MAP4K4EGFRFRKCSNK1A1
SCHEMBL29640899 0.77 LATS1 (0.37) MAPK9MAP4K4EGFRFRKCSNK1A1
SCHEMBL26289615 0.76 MEN1 (0.37) MAP4K4RPS6KA5RPS6KA4MAPTMEN1
SCHEMBL30438289 0.76 MEN1 (0.37) MAP4K4RPS6KA5RPS6KA4MAPTMEN1
SCHEMBL29627704 0.74 HSP90AA1 (0.42) MAPK9MAPK14RPS6KA5MAPK10GRM5
SCHEMBL6449580 0.74 HSP90AA1 (0.42) MAPK9MAPK14RPS6KA5MAPK10GRM5
SCHEMBL6101938 0.74 KDM4E (0.59) MAPTKMT2AGRM5HSP90AA1ALDH1A1
SCHEMBL2650448 0.74 L3MBTL1 (0.49) MAPTMEN1KMT2AALDH1A1NPC1
SCHEMBL30061028 0.74 L3MBTL1 (0.49) MAPTMEN1KMT2AALDH1A1NPC1
SCHEMBL30620644 0.73 NPC1 (0.47) RPS6KA5RPS6KA4KMT2AGRM5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed