SCHEMBL29643377

SCHEMBL29643377

Cc1ccc(C#Cc2ccccc2)c([N+](=O)[O-])c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.51
CYP3A4 P08684 1/20 0.51
CASP3 P42574 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
HSD17B10 Q99714 1/20 0.41
KCNMA1 Q12791 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 1/20 0.40
GPR35 Q9HC97 1/20 0.40
ALDH1A1 P00352 4/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
ACHE P22303 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
CA12 O43570 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19063495 1.00 TSHR (0.51) TSHRCYP3A4CASP3SENP8SENP7
SCHEMBL4460747 0.84 TSHR (0.45) TSHRCYP3A4ALDH1A1
SCHEMBL12984706 0.84 TSHR (0.46) TSHRCYP3A4CASP3SENP8SENP7
SCHEMBL19622953 0.83 CASP3 (0.53) TSHRCYP3A4CASP3SENP8SENP7
SCHEMBL28923654 0.83 HSD17B10 (0.46) TSHRCYP3A4CASP3SENP8SENP7
SCHEMBL28623382 0.81 ATM (0.46) CYP3A4CASP3SENP8SENP7SENP6
SCHEMBL29669613 0.81 VCAM1 (0.59) TSHRCYP3A4CASP3SENP8SENP7
SCHEMBL28487454 0.81 CA12 (0.50) TSHRCYP3A4CASP3SENP8SENP7
SCHEMBL3421225 0.81 CASP3 (0.44) TSHRCYP3A4CASP3SENP8SENP7
SCHEMBL28641030 0.81 RAB9A (0.49) NPC1RAB9AALDH1A1CA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429424-B Preparation method of [1,2,4] oxadiazino indoline-3-ketone derivative 华侨大学 2022-06-07 CN claimed
CN-113429424-B Preparation method of [1,2,4] oxadiazino indoline-3-ketone derivative 华侨大学 2022-06-07 CN disclosed