SCHEMBL29644336

SCHEMBL29644336

COc1ccc(C(=O)N2CCc3c(cccc3C(CC(=O)O)c3ccccc3)C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.50
KMT2A Q03164 2/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
USP2 O75604 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
PRMT5 O14744 3/20 0.46
WDR77 Q9BQA1 3/20 0.46
NAMPT P43490 2/20 0.46
DRD4 P21917 1/20 0.46
ALDH1A1 P00352 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MEN1 O00255 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.44
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
RAB9A P51151 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28739159 1.00 FFAR1 (0.50) FFAR1KMT2ALMNAMAPTHPGD
SCHEMBL28739082 0.97 FFAR1 (0.51) FFAR1KMT2ALMNAMAPTHPGD
SCHEMBL29644457 0.97 FFAR1 (0.51) FFAR1KMT2ALMNAMAPTHPGD
SCHEMBL28739120 0.91 FFAR1 (0.48) FFAR1KMT2ALMNAMAPTHPGD
SCHEMBL29644442 0.91 FFAR1 (0.48) FFAR1KMT2ALMNAMAPTHPGD
SCHEMBL29644389 0.90 LMNA (0.49) FFAR1KMT2ALMNAMAPTHPGD
SCHEMBL28739096 0.90 LMNA (0.49) FFAR1KMT2ALMNAMAPTHPGD
SCHEMBL29644422 0.90 FFAR1 (0.49) FFAR1KMT2ALMNAMAPTHPGD
SCHEMBL29644419 0.90 NFE2L2 (0.49) FFAR1LMNAHPGDCYP3A4CYP2D6
SCHEMBL28739160 0.90 NFE2L2 (0.49) FFAR1LMNAHPGDCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114507181-B Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-03-26 CN disclosed
CN-114507181-A Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-05-17 CN disclosed