SCHEMBL29644422

SCHEMBL29644422

COc1ccc(C(=O)N2CCc3c(cccc3C(CC(=O)O)c3ccc(C#N)cc3)C2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 3/20 0.49
USP2 O75604 5/20 0.44
TSHR P16473 5/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PTGER4 P35408 1/20 0.43
PTGER2 P43116 1/20 0.43
PTGDR Q13258 1/20 0.43
CYP3A4 P08684 5/20 0.43
CYP2D6 P10635 1/20 0.43
GRM5 P41594 2/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
HPGD P15428 2/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.42
DRD4 P21917 1/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28739128 1.00 FFAR1 (0.49) FFAR1USP2TSHRCYP1A2CYP2C9
SCHEMBL28739066 0.93 FFAR1 (0.44) FFAR1USP2TSHRCYP1A2CYP2C9
SCHEMBL29644332 0.93 FFAR1 (0.44) FFAR1USP2TSHRCYP1A2CYP2C9
SCHEMBL29644457 0.93 FFAR1 (0.51) FFAR1USP2CYP2C9CYP3A4CYP2D6
SCHEMBL28739082 0.93 FFAR1 (0.51) FFAR1USP2CYP2C9CYP3A4CYP2D6
SCHEMBL28739159 0.90 FFAR1 (0.50) FFAR1USP2CYP2C9SMN1; SMN2CYP3A4
SCHEMBL29644336 0.90 FFAR1 (0.50) FFAR1USP2CYP2C9SMN1; SMN2CYP3A4
SCHEMBL28739096 0.86 LMNA (0.49) FFAR1MAPTKMT2AHPGDALDH1A1
SCHEMBL29644389 0.86 LMNA (0.49) FFAR1MAPTKMT2AHPGDALDH1A1
SCHEMBL29644431 0.85 MAPK1 (0.48) FFAR1TSHRMAPTKMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114507181-B Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-03-26 CN disclosed
CN-114507181-A Propionic acid compound containing 5-substituted tetrahydroisoquinoline, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-05-17 CN disclosed