SCHEMBL29645656

SCHEMBL29645656

COc1ccc(-c2nc3c4c(N5CCOCC5)cccc4nc(Nc4ccccnc4=O)n3n2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.44
CASP1 P29466 6/20 0.39
CASP7 P55210 6/20 0.39
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
USP2 O75604 5/20 0.39
TSHR P16473 3/20 0.39
MAPT P10636 3/20 0.39
THRB P10828 1/20 0.39
ALDH1A1 P00352 8/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP1A2 P05177 5/20 0.38
HSD17B10 Q99714 4/20 0.38
LMNA P02545 2/20 0.38
HIF1A Q16665 3/20 0.38
PIK3CD O00329 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29645455 0.88 PIK3CA (0.42) PIK3CACASP1CASP7MEN1KMT2A
SCHEMBL29645530 0.85 PDE10A (0.42) PIK3CACASP1CASP7MEN1KMT2A
SCHEMBL29645863 0.84 MAPT (0.44) MAPTTHRBALDH1A1KDM4ESMN1; SMN2
SCHEMBL29645660 0.84 MAPT (0.44) MAPTTHRBALDH1A1KDM4EGAA
SCHEMBL29646084 0.84 MAPT (0.40) PIK3CACASP1CASP7MEN1KMT2A
SCHEMBL29645991 0.83 MAPT (0.44) MAPTTHRBALDH1A1KDM4ESMN1; SMN2
SCHEMBL29645468 0.83 MAPT (0.44) KMT2AMAPTTHRBALDH1A1KDM4E
SCHEMBL29645567 0.82 MAPT (0.41) CASP1CASP7MEN1KMT2AUSP2
SCHEMBL29646050 0.81 MAPT (0.42) MEN1KMT2AMAPTTHRBALDH1A1
SCHEMBL29645487 0.81 MAPT (0.59) MAPTTHRBALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN disclosed