SCHEMBL29646286

SCHEMBL29646286

c1ccc(Cn2c(NCc3ccco3)nc3ccccc32)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPC5 Q9UL62 7/20 1.00
TRPC4 Q9UBN4 2/20 1.00
SMN1; SMN2 Q16637 2/20 0.70
HTT P42858 1/20 0.70
USP2 O75604 1/20 0.67
MAPK1 P28482 1/20 0.67
ALDH1A1 P00352 1/20 0.65
MAPT P10636 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22619593 1.00 TRPC5 (1.00) TRPC5TRPC4SMN1; SMN2HTTUSP2
SCHEMBL1170660 0.85 ALDH1A1 (0.86) TRPC5TRPC4SMN1; SMN2HTTALDH1A1
SCHEMBL20715328 0.82 SMN1; SMN2 (1.00) TRPC5TRPC4SMN1; SMN2HTTUSP2
SCHEMBL19714457 0.81 TSHR (0.71) TRPC5TRPC4SMN1; SMN2HTTUSP2
SCHEMBL1170123 0.76 SMN1; SMN2 (0.74) TRPC5TRPC4SMN1; SMN2HTTALDH1A1
SCHEMBL1169982 0.75 ALDH1A1 (0.69) TRPC5TRPC4SMN1; SMN2HTTMAPK1
SCHEMBL28805359 0.73 MAPT (0.62) TRPC5TRPC4SMN1; SMN2HTTALDH1A1
Hydrochloric Acid SCHEMBL28745357 0.73 CYP1A2 (0.66) TRPC5TRPC4SMN1; SMN2HTTALDH1A1
SCHEMBL1170308 0.72 ALDH1A1 (0.61) TRPC5TRPC4SMN1; SMN2ALDH1A1MAPT
SCHEMBL1170118 0.71 KMT2A (0.64) TRPC5TRPC4SMN1; SMN2HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114642744-B Method for screening morphine-tolerance-relieving drugs 南京医科大学 2023-05-23 CN disclosed
CN-114642744-A Method for screening morphine tolerance relieving drugs 南京医科大学 2022-06-21 CN disclosed