SCHEMBL29647640

SCHEMBL29647640

O=C1C(c2ccc(F)cc2)=CC(=O)c2c(O)cccc21

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 7/20 0.78
AURKA O14965 2/20 0.58
DYRK1A Q13627 1/20 0.58
MAPT P10636 5/20 0.54
KDM4E B2RXH2 4/20 0.54
RECQL P46063 4/20 0.54
ALDH1A1 P00352 3/20 0.54
HPGD P15428 3/20 0.54
ALOX15 P16050 3/20 0.54
MAPK1 P28482 3/20 0.54
HSD17B10 Q99714 3/20 0.54
TDP1 Q9NUW8 3/20 0.54
KMT2A Q03164 3/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
MEN1 O00255 2/20 0.54
TRPA1 O75762 2/20 0.54
TP53 P04637 2/20 0.54
CYP3A4 P08684 2/20 0.54
CASP1 P29466 2/20 0.54
CDC25B P30305 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27006529 1.00 BACE1 (0.78) BACE1AURKADYRK1AMAPTKDM4E
SCHEMBL14305571 0.88 BACE1 (1.00) BACE1AURKADYRK1AMAPTKDM4E
SCHEMBL24389333 0.86 BACE1 (1.00) BACE1AURKADYRK1AMAPTKDM4E
SCHEMBL29647664 0.81 BACE1 (0.73) BACE1AURKADYRK1AMAPTKDM4E
SCHEMBL27006528 0.81 BACE1 (0.73) BACE1AURKADYRK1AMAPTKDM4E
SCHEMBL28339368 0.77 BACE1 (0.72) BACE1MAPTALDH1A1HPGDMAPK1
SCHEMBL1042858 0.76 BACE1 (0.81) BACE1AURKADYRK1AMAPTKDM4E
SCHEMBL8652779 0.75 CASP3 (0.57) BACE1AURKADYRK1AMAPTKDM4E
SCHEMBL29647621 0.75 GAPDH (0.77) BACE1AURKADYRK1AMAPTKDM4E
SCHEMBL27006543 0.75 GAPDH (0.77) BACE1AURKADYRK1AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4232439-A1 5-HYDROXY-1,4-NAPHTHALENEDIONE FOR USE IN THE TREATMENT OF CANCER Godavari Biorefineries Ltd. (IN) 2023-08-30 EP disclosed
CN-116670122-A 5-hydroxy-1, 4-naphthalenediones for the treatment of cancer 戈达瓦里生物炼制有限责任公司 2023-08-29 CN disclosed
WO-2022091123-A1 5-HYDROXY-1,4-NAPHTHALENEDIONE FOR USE IN THE TREATMENT OF CANCER GODAVARI BIOREFINERIES LIMITED (IN) 2022-05-05 WO disclosed