SCHEMBL29650673

SCHEMBL29650673

Brc1cc(-c2ccncc2)cc2cnccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCD Q05655 9/20 0.51
PRKCH P24723 8/20 0.51
PRKCE Q02156 8/20 0.51
PRKCQ Q04759 8/20 0.51
LATS1 O95835 1/20 0.47
LATS2 Q9NRM7 1/20 0.47
PIM1 P11309 2/20 0.42
HASPIN Q8TF76 2/20 0.42
CCNT1 O60563 1/20 0.42
CDK9 P50750 1/20 0.42
PRKCZ Q05513 2/20 0.42
PRKD2 Q9BZL6 1/20 0.42
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
IMPDH2 P12268 1/20 0.41
PRKCA P17252 4/20 0.40
PRKCB P05771 3/20 0.40
PRKD1 Q15139 2/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3324615 1.00 PRKCD (0.51) PRKCDPRKCHPRKCEPRKCQLATS1
SCHEMBL30855724 0.79 IMPDH2 (0.44) PRKCDPRKCHPRKCEPRKCQPIM1
SCHEMBL21201370 0.79 IMPDH2 (0.44) PRKCDPRKCHPRKCEPRKCQPIM1
SCHEMBL3326564 0.78 PRKCH (0.55) PRKCDPRKCHPRKCEPRKCQLATS1
SCHEMBL15488451 0.77 IMPDH2 (0.43) PIM1HASPINCCNT1CDK9LMNA
SCHEMBL3327006 0.74 PRKCD (0.56) PRKCDPRKCHPRKCEPRKCQLATS1
SCHEMBL3713151 0.74 MAPK10 (0.48) PIM1HASPINCCNT1CDK9PRKCZ
SCHEMBL21917154 0.73 CHUK (0.44) PIM1HASPINCCNT1CDK9IMPDH2
SCHEMBL23301129 0.72 PRKCZ (0.43) PRKCDPRKCHPRKCEPRKCQPIM1
SCHEMBL23328129 0.72 PDE2A (0.40) PRKCDPRKCHPRKCEPRKCQPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114621222-B 6-6 Fused bicyclic heteroaryl compounds and their use as LATS inhibitors 诺华股份有限公司 2024-12-17 CN disclosed
CN-110573511-B 6-6 fused bicyclic heteroaryl compounds and their use as LATS inhibitors 诺华股份有限公司 2023-04-25 CN disclosed
CN-114703144-A 6-6 fused bicyclic heteroaryl compounds and their use as LATS inhibitors 诺华股份有限公司 2022-07-05 CN disclosed
CN-114621222-A 6-6 fused bicyclic heteroaryl compounds and their use as LATS inhibitors 诺华股份有限公司 2022-06-14 CN disclosed