SCHEMBL29655165

SCHEMBL29655165

COc1cc(F)ccc1-c1ccc(N)c([N+](=O)[O-])c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 6/20 0.54
MAPT P10636 5/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
POLB P06746 1/20 0.54
HTT P42858 2/20 0.46
TSHR P16473 1/20 0.44
ALDH1A1 P00352 4/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX15 P16050 1/20 0.43
ABCB1 P08183 2/20 0.42
ABCC1 P33527 2/20 0.42
NPSR1 Q6W5P4 1/20 0.41
GALR3 O60755 1/20 0.41
THRB P10828 1/20 0.41
S1PR1 P21453 1/20 0.41
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
RECQL P46063 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29655083 0.85 TDP1 (0.55) TDP1MAPTMEN1KMT2APOLB
SCHEMBL29655065 0.85 TDP1 (0.58) TDP1MAPTMEN1KMT2APOLB
SCHEMBL5952257 0.85 TDP1 (0.58) TDP1MAPTMEN1KMT2APOLB
SCHEMBL11688979 0.82 ADORA3 (0.51) TDP1MEN1KMT2AHTTPDGFRB
SCHEMBL29655271 0.82 TDP1 (0.62) TDP1MAPTMEN1KMT2APOLB
SCHEMBL29655054 0.80 TDP1 (0.47) TDP1MEN1KMT2ATSHRALDH1A1
SCHEMBL29655119 0.79 MAPT (0.54) TDP1MAPTMEN1KMT2APOLB
SCHEMBL29655063 0.79 TDP1 (0.54) TDP1MAPTMEN1KMT2APOLB
SCHEMBL18985825 0.78 MAPT (0.53) TDP1MAPTMEN1KMT2APOLB
SCHEMBL720358 0.77 TDP1 (0.79) TDP1MAPTMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843874-B Phthalazine derivatives useful as inhibitors of PARP1, PARP2 and/or tubulin for the treatment of cancer 加利福尼亚大学董事会 2022-05-27 CN disclosed