SCHEMBL29655271

SCHEMBL29655271

Nc1ccc(-c2ccc(F)cc2F)cc1[N+](=O)[O-]

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.62
MAPT P10636 4/20 0.62
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
POLB P06746 2/20 0.62
ATM Q13315 1/20 0.53
ALDH1A1 P00352 5/20 0.49
CYP3A4 P08684 1/20 0.49
ALOX15 P16050 1/20 0.49
TSHR P16473 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSPB1 P04792 2/20 0.43
LMNA P02545 2/20 0.43
HIF1A Q16665 2/20 0.42
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
DHFR P00374 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
TTR P02766 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27963778 0.88 ALDH1A1 (0.62) TDP1MAPTMEN1KMT2APOLB
SCHEMBL2654089 0.86 TDP1 (0.58) TDP1MAPTMEN1KMT2APOLB
SCHEMBL29655079 0.83 TDP1 (0.64) TDP1MAPTMEN1KMT2APOLB
SCHEMBL719169 0.83 TDP1 (0.64) TDP1MAPTMEN1KMT2APOLB
SCHEMBL720358 0.82 TDP1 (0.79) TDP1MAPTMEN1KMT2APOLB
SCHEMBL29655119 0.82 MAPT (0.54) TDP1MAPTMEN1KMT2APOLB
SCHEMBL29655165 0.82 TDP1 (0.54) TDP1MAPTMEN1KMT2APOLB
SCHEMBL15156399 0.82 MAPT (0.54) TDP1MAPTMEN1KMT2APOLB
SCHEMBL537892 0.82 TDP1 (0.64) TDP1MAPTMEN1KMT2APOLB
SCHEMBL9808951 0.80 TDP1 (0.55) TDP1MAPTMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843874-B Phthalazine derivatives useful as inhibitors of PARP1, PARP2 and/or tubulin for the treatment of cancer 加利福尼亚大学董事会 2022-05-27 CN disclosed