SCHEMBL29658484

SCHEMBL29658484

CCc1c(C#N)c(S)nc(N2CCC(N3CCCC3)CC2)c1C#N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.41
KDM4E B2RXH2 9/20 0.41
HPGD P15428 7/20 0.41
GAA P10253 4/20 0.41
DNMT1 P26358 1/20 0.39
PDCD1 Q15116 2/20 0.38
CD274 Q9NZQ7 2/20 0.38
MAPT P10636 1/20 0.38
HRH3 Q9Y5N1 4/20 0.37
HSD17B10 Q99714 2/20 0.36
HIF1A Q16665 2/20 0.36
RECQL P46063 1/20 0.36
POLB P06746 2/20 0.36
LMNA P02545 3/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
L3MBTL3 Q96JM7 1/20 0.34
HTT P42858 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19717166 1.00 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDGAADNMT1
SCHEMBL19734832 0.87 ALDH1A1 (0.52) ALDH1A1KDM4EHPGDGAAMAPT
SCHEMBL19717353 0.85 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDGAADNMT1
SCHEMBL29658627 0.85 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDGAADNMT1
SCHEMBL19734994 0.84 DNMT1 (0.53) ALDH1A1KDM4EHPGDGAADNMT1
SCHEMBL19734950 0.81 DNMT1 (0.40) ALDH1A1KDM4EHPGDGAADNMT1
SCHEMBL19717302 0.80 DNMT1 (0.38) ALDH1A1KDM4EHPGDGAADNMT1
SCHEMBL29658560 0.80 DNMT1 (0.38) ALDH1A1KDM4EHPGDGAADNMT1
SCHEMBL19734861 0.79 KDM4E (0.49) ALDH1A1KDM4EHPGDGAADNMT1
SCHEMBL19734698 0.78 KDM4E (0.54) ALDH1A1KDM4EHPGDMAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563043-B Substituted pyridines as inhibitors of DNMT1 葛兰素史密斯克莱知识产权发展有限公司 2022-05-31 CN disclosed