SCHEMBL29658554

SCHEMBL29658554

NC(=O)C(O)c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
MAPT P10636 2/20 0.45
HTT P42858 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GABBR2 O75899 3/20 0.44
GABBR1 Q9UBS5 3/20 0.44
LMNA P02545 3/20 0.44
CYP2C9 P11712 3/20 0.44
TSHR P16473 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CYP3A4 P08684 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
NFKB1 P19838 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19717863 1.00 BRD4 (0.45) BRD4HDAC4HDAC7HDAC5MAPT
SCHEMBL5068690 1.00 BRD4 (0.45) BRD4HDAC4HDAC7HDAC5MAPT
SCHEMBL5068688 1.00 BRD4 (0.45) BRD4HDAC4HDAC7HDAC5MAPT
SCHEMBL29386802 0.81 BRD4 (0.48) BRD4HDAC4HDAC7HDAC5MAPT
SCHEMBL22082538 0.79 LMNA (0.39) MAPTSMN1; SMN2LMNACYP2C9TSHR
SCHEMBL22082536 0.79 LMNA (0.39) MAPTSMN1; SMN2LMNACYP2C9TSHR
SCHEMBL6367 0.79 LMNA (0.62) BRD4HDAC4HDAC7HDAC5NPSR1
SCHEMBL20853599 0.79 BRD4 (0.47) BRD4HDAC4HDAC7HDAC5MAPT
SCHEMBL22081099 0.79 LMNA (0.39) MAPTSMN1; SMN2LMNACYP2C9TSHR
SCHEMBL6366 0.79 LMNA (0.62) BRD4HDAC4HDAC7HDAC5NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563043-B Substituted pyridines as inhibitors of DNMT1 葛兰素史密斯克莱知识产权发展有限公司 2022-05-31 CN disclosed