SCHEMBL29658592

SCHEMBL29658592

NC(=O)C(O)c1ccc(F)nc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.36
P2RX7 Q99572 2/20 0.34
FOLH1 Q04609 1/20 0.34
KCNQ3 O43525 1/20 0.33
KCNQ2 O43526 1/20 0.33
MET P08581 1/20 0.33
MST1R Q04912 1/20 0.33
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
F10 P00742 1/20 0.32
BTK Q06187 1/20 0.31
APLNR P35414 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2A6 P11509 1/20 0.31
CYP2B6 P20813 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19716584 1.00 EPHX2 (0.36) EPHX2P2RX7FOLH1KCNQ3KCNQ2
SCHEMBL2761040 0.80 P2RX7 (0.37) P2RX7METMST1RAPLNR
SCHEMBL2760832 0.77 TRPV4 (0.43) P2RX7CES2CES1
SCHEMBL19544649 0.76 CYP2A6 (0.36) EPHX2P2RX7FOLH1KCNQ3KCNQ2
SCHEMBL4092644 0.74 HDAC3 (0.45) CES2CES1
SCHEMBL19735013 0.74 HDAC3 (0.45) CES2CES1
SCHEMBL3554668 0.73 EPHX2 (0.41) EPHX2P2RX7FOLH1KCNQ3KCNQ2
SCHEMBL19716738 0.73 LOXL2 (0.39) METMST1RCES2CES1F10
SCHEMBL29658521 0.73 LOXL2 (0.39) METMST1RCES2CES1F10
SCHEMBL19716826 0.73 FOLH1 (0.32) EPHX2P2RX7FOLH1APLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563043-B Substituted pyridines as inhibitors of DNMT1 葛兰素史密斯克莱知识产权发展有限公司 2022-05-31 CN disclosed