SCHEMBL29665255

SCHEMBL29665255

Oc1cnnc2ccc(Br)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.39
CASP1 P29466 2/20 0.37
GAA P10253 1/20 0.37
CASP7 P55210 1/20 0.37
ALK Q9UM73 1/20 0.37
ERN1 O75460 1/20 0.37
BCL2 P10415 1/20 0.36
MCL1 Q07820 1/20 0.36
PIM1 P11309 2/20 0.36
CHEK1 O14757 1/20 0.36
AKT1 P31749 1/20 0.36
FLT3 P36888 1/20 0.36
PIM3 Q86V86 1/20 0.36
HTT P42858 1/20 0.36
PABPC1 P11940 1/20 0.35
IDO1 P14902 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
EGFR P00533 1/20 0.35
CES2 O00748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL796509 1.00 ALOX15 (0.39) ALOX15CASP1GAACASP7ALK
SCHEMBL16294313 0.85 ALOX15 (0.39) ALOX15CASP1ERN1BCL2MCL1
Hydrochloric Acid SCHEMBL29015486 0.83 ALOX15 (0.38) ALOX15CASP1ERN1BCL2MCL1
SCHEMBL12861090 0.77 SRC (0.32)
SCHEMBL4297621 0.77 NT5E (0.49) GAAALKPIM1CHEK1AKT1
SCHEMBL30950664 0.77 NT5E (0.49) GAAALKPIM1CHEK1AKT1
SCHEMBL29665280 0.77 NT5E (0.49) GAAALKPIM1CHEK1AKT1
SCHEMBL12034330 0.77 TRPA1 (0.45) ALOX15GAAIDO1LMNAMAPT
SCHEMBL9998167 0.77 ERN1 (0.37) ERN1
SCHEMBL2719952 0.77 KDM4E (0.44) HTTIDO1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118388416-A Synthesis method of 4-chloro-6-bromocinnoline 凯美克(上海)医药科技有限公司 2024-07-26 CN claimed
CN-118388416-A Synthesis method of 4-chloro-6-bromocinnoline 凯美克(上海)医药科技有限公司 2024-07-26 CN disclosed
CN-118388416-A Synthesis method of 4-chloro-6-bromocinnoline 凯美克(上海)医药科技有限公司 2024-07-26 CN disclosed
EP-4251617-A1 (AZA)QUINOLINE 4-AMINES DERIVATIVES AS P2X3 INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2023-10-04 EP disclosed
WO-2022112491-A1 (AZA)QUINOLINE 4-AMINES DERIVATIVES AS P2X3 INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2022-06-02 WO disclosed