SCHEMBL796509

SCHEMBL796509

Oc1cnnc2ccc(Br)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.39
CASP1 P29466 2/20 0.37
GAA P10253 1/20 0.37
CASP7 P55210 1/20 0.37
ALK Q9UM73 1/20 0.37
ERN1 O75460 1/20 0.37
BCL2 P10415 1/20 0.36
MCL1 Q07820 1/20 0.36
PIM1 P11309 2/20 0.36
CHEK1 O14757 1/20 0.36
AKT1 P31749 1/20 0.36
FLT3 P36888 1/20 0.36
PIM3 Q86V86 1/20 0.36
HTT P42858 1/20 0.36
PABPC1 P11940 1/20 0.35
IDO1 P14902 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
EGFR P00533 1/20 0.35
CES2 O00748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29665255 1.00 ALOX15 (0.39) ALOX15CASP1GAACASP7ALK
SCHEMBL16294313 0.85 ALOX15 (0.39) ALOX15CASP1ERN1BCL2MCL1
Hydrochloric Acid SCHEMBL29015486 0.83 ALOX15 (0.38) ALOX15CASP1ERN1BCL2MCL1
SCHEMBL12861090 0.77 SRC (0.32)
SCHEMBL4297621 0.77 NT5E (0.49) GAAALKPIM1CHEK1AKT1
SCHEMBL30950664 0.77 NT5E (0.49) GAAALKPIM1CHEK1AKT1
SCHEMBL29665280 0.77 NT5E (0.49) GAAALKPIM1CHEK1AKT1
SCHEMBL12034330 0.77 TRPA1 (0.45) ALOX15GAAIDO1LMNAMAPT
SCHEMBL9998167 0.77 ERN1 (0.37) ERN1
SCHEMBL2719952 0.77 KDM4E (0.44) HTTIDO1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250213571-A1 TYK2 INHIBITORS AND USES THEREOF ALUMIS INC. 2025-07-03 US disclosed
EP-4493562-A1 TYK2 INHIBITORS AND USES THEREOF Alumis Inc. (US) 2025-01-22 EP disclosed
CN-118388416-A Synthesis method of 4-chloro-6-bromocinnoline 凯美克(上海)医药科技有限公司 2024-07-26 CN disclosed
US-20240207263-A1 SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF SUZHOU ZANRONG PHARMA LIMITED (CN) 2024-06-27 US disclosed
EP-4308569-A1 SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF Suzhou Zanrong Pharma Limited (CN) 2024-01-24 EP disclosed
CN-117412972-A Selective modulators of Ataxia Telangiectasia Mutated (ATM) kinase and uses thereof 苏州赞荣医药科技有限公司 2024-01-16 CN disclosed
WO-2023178235-A1 TYK2 INHIBITORS AND USES THEREOF ALUMIS INC. (US) 2023-09-21 WO disclosed
WO-2023178235-A1 TYK2 INHIBITORS AND USES THEREOF ALUMIS INC. (US) 2023-09-21 WO disclosed
WO-2022193166-A1 SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF SUZHOU ZANRONG PHARMA LIMITED (CN) 2022-09-22 WO disclosed
WO-2022194138-A1 SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF SUZHOU ZANRONG PHARMA LIMITED (CN) 2022-09-22 WO disclosed
US-9181264-B2 Fused heteroaryls and their uses HUTCHISON MEDIPHARMA LIMITED (CN) 2015-11-10 US disclosed
US-9181264-B2 Fused heteroaryls and their uses HUTCHISON MEDIPHARMA LIMITED (CN) 2015-11-10 US disclosed
US-20130190307-A1 FUSED HETEROARYLS AND THEIR USES HUTCHISON MEDIPHARMA LIMITED (CN) 2013-07-25 US disclosed
US-20130190307-A1 FUSED HETEROARYLS AND THEIR USES HUTCHISON MEDIPHARMA LIMITED (CN) 2013-07-25 US disclosed
US-20130190307-A1 FUSED HETEROARYLS AND THEIR USES HUTCHISON MEDIPHARMA LIMITED (CN) 2013-07-25 US disclosed
EP-2616468-A1 FUSED HETEROARYLS AND THEIR USES Hutchison Medipharma Limited (CN) 2013-07-24 EP disclosed
CN-103124731-A Fused heteroaryl compounds and uses thereof HUTCHISON MEDIPHARMA LTD 2013-05-29 CN disclosed
CN-102399218-A Triheterocyclic compounds and their use as PI3K inhibitors HUTCHISON MEDIPHARMA LTD 2012-04-04 CN disclosed
WO-2012034526-A1 FUSED HETEROARYLS AND THEIR USES HUTCHISON MEDIPHARMA LIMITED (CN) 2012-03-22 WO disclosed
WO-2012034526-A1 FUSED HETEROARYLS AND THEIR USES HUTCHISON MEDIPHARMA LIMITED (CN) 2012-03-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250213571-A1 TYK2 INHIBITORS AND USES THEREOF TYK2, JAK1, JAK2 ALOX15 1980/4885CASP1 1831/4885GAA 3318/4885
US-20130190307-A1 FUSED HETEROARYLS AND THEIR USES FARS2, TIAL1, DHFR ALOX15 2675/4885CASP1 2297/4885GAA 2258/4885
US-20240207263-A1 SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF ATM, CHEK2, CHEK1 ALOX15 4651/4885CASP1 2793/4885GAA 485/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.