SCHEMBL29665264

SCHEMBL29665264

CC(C)(C)OC(=O)N1CCN(c2ccc(N)cc2C#N)CC1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.54
GAA P10253 1/20 0.54
HSD17B10 Q99714 1/20 0.54
NR1H2 P55055 2/20 0.51
SMARCA2 P51531 1/20 0.48
SMARCA4 P51532 1/20 0.48
PBRM1 Q86U86 1/20 0.48
GPR119 Q8TDV5 5/20 0.48
LMNA P02545 2/20 0.46
NR1H3 Q13133 1/20 0.46
ALDH1A1 P00352 1/20 0.45
RET P07949 3/20 0.45
EGLN2 Q96KS0 1/20 0.45
MAP4K4 O95819 1/20 0.44
PIK3CA P42336 1/20 0.43
BACE1 P56817 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL594432 1.00 MAPT (0.54) MAPTGAAHSD17B10NR1H2SMARCA2
SCHEMBL6052351 0.95 MAPT (0.50) MAPTGAAHSD17B10NR1H2SMARCA2
SCHEMBL6052124 0.89 IRAK4 (0.47) MAPTGAAHSD17B10NR1H2GPR119
SCHEMBL23220924 0.86 MEN1 (0.49) MAPTNR1H2GPR119LMNANR1H3
SCHEMBL652725 0.85 MEN1 (0.52) MAPTNR1H2GPR119LMNANR1H3
SCHEMBL28744864 0.85 MAPT (0.54) MAPTGAAHSD17B10LMNAALDH1A1
SCHEMBL2459991 0.85 GPR119 (0.50) MAPTNR1H2GPR119LMNANR1H3
SCHEMBL355300 0.85 BACE1 (0.55) MAPTNR1H2GPR119LMNANR1H3
SCHEMBL2462125 0.84 ALDH1A1 (0.51) MAPTGAAHSD17B10NR1H2GPR119
SCHEMBL25403559 0.83 SMARCA2 (0.47) MAPTNR1H2SMARCA2SMARCA4PBRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113651799-B Six-membered non-aromatic ring-containing diaryl pyrimidine HIV-1 reverse transcriptase inhibitor and preparation method and application thereof 山东大学 2022-06-17 CN claimed
CN-118742539-A Heterocyclic derivative and preparation method and application thereof 浙江海正药业股份有限公司 2024-10-01 CN disclosed
CN-113651799-B Six-membered non-aromatic ring-containing diaryl pyrimidine HIV-1 reverse transcriptase inhibitor and preparation method and application thereof 山东大学 2022-06-17 CN disclosed