SCHEMBL29671111

SCHEMBL29671111

COC(=O)[C@@H](N)Cc1ccc(Br)c2nccnc12

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.35
ALDH1A1 P00352 1/20 0.35
IDO1 P14902 1/20 0.31
HDAC6 Q9UBN7 4/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
HDAC1 Q13547 2/20 0.31
LTA4H P09960 2/20 0.31
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2C Q14957 1/20 0.31
POLB P06746 1/20 0.31
KIF11 P52732 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28572795 1.00 PTGS2 (0.35) PTGS2ALDH1A1IDO1HDAC6MEN1
SCHEMBL22031968 0.85 KMT2A (0.45) PTGS2ALDH1A1MEN1KMT2A
SCHEMBL29579589 0.85 KDM4E (0.41) PTGS2ALDH1A1MEN1KMT2A
SCHEMBL29671158 0.85 KMT2A (0.45) PTGS2ALDH1A1MEN1KMT2A
SCHEMBL28574369 0.84 PTGS2 (0.35) PTGS2ALDH1A1HDAC6HDAC1GRIN3B
Hydrochloric Acid SCHEMBL29671147 0.84 KMT2A (0.45) PTGS2ALDH1A1MEN1KMT2A
SCHEMBL29671089 0.84 PTGS2 (0.35) PTGS2ALDH1A1HDAC6HDAC1GRIN3B
SCHEMBL21979243 0.83 HSD17B10 (0.42) ALDH1A1MEN1KMT2AGRIN3BGRIN1
SCHEMBL21979244 0.83 HSD17B10 (0.42) ALDH1A1MEN1KMT2AGRIN3BGRIN1
Hydrochloric Acid SCHEMBL30901269 0.83 HDAC8 (0.34) PTGS2ALDH1A1HDAC6HDAC1GRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3873605-B1 COMPOUNDS FOR INHIBITION OF ALPHA4BETA7 INTEGRIN GILEAD SCIENCES INC (US) 2024-10-23 EP disclosed
US-20220152014-A1 COMPOUNDS FOR INHIBITION OF ALPHA 4 BETA 7 INTEGRIN GILEAD SCIENCES, INC. (US) 2022-05-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220152014-A1 COMPOUNDS FOR INHIBITION OF ALPHA 4 BETA 7 INTEGRIN ITGB7, ITGB4, ITGA4 PTGS2 2563/4885ALDH1A1 823/4885IDO1 4608/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.