SCHEMBL29673141

SCHEMBL29673141

CC(C)(C)OC(=O)N1CCN(c2nc(Cl)nc(CBr)c2[N+](=O)[O-])CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.48
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
POLB P06746 1/20 0.38
CCNT1 O60563 1/20 0.37
CDK9 P50750 1/20 0.37
GBA1 P04062 2/20 0.36
ABL1 P00519 1/20 0.36
BCR P11274 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
CKS1B P61024 1/20 0.36
SKP1 P63208 1/20 0.36
SKP2 Q13309 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TLR9 Q9NR96 1/20 0.36
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28766422 1.00 KCNH2 (0.48) KCNH2ALDH1A1LMNAMAPTPOLB
SCHEMBL29673158 0.85 MAPT (0.50) KCNH2ALDH1A1LMNAMAPTPOLB
SCHEMBL28768664 0.85 MAPT (0.50) KCNH2ALDH1A1LMNAMAPTPOLB
SCHEMBL28766498 0.84 GPR119 (0.41) KCNH2ALDH1A1LMNAMAPTGPR119
SCHEMBL28766492 0.84 GPR119 (0.41) KCNH2ALDH1A1LMNAMAPTGPR119
SCHEMBL29673070 0.84 GPR119 (0.41) KCNH2ALDH1A1LMNAMAPTGPR119
SCHEMBL29724314 0.83 ABL1 (0.42) ALDH1A1LMNAMAPTABL1BCR
SCHEMBL20213112 0.82 KCNH2 (0.48) KCNH2ALDH1A1LMNAMAPTPOLB
SCHEMBL1693887 0.76 ALDH1A1 (0.44) KCNH2ALDH1A1LMNAMAPTCCNT1
SCHEMBL6628480 0.75 MAPT (0.52) KCNH2ALDH1A1LMNAMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022127827-A1 KRASG12C PROTEIN MUTATION INHIBITOR AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 上海维申医药有限公司 2022-06-23 WO disclosed
CN-114644631-A KRAS G12C protein mutation inhibitor, preparation method thereof, pharmaceutical composition and application thereof 上海维申医药有限公司 2022-06-21 CN disclosed