SCHEMBL29675587

SCHEMBL29675587

CC(=O)N[C@H](C)c1cc(F)cc(N2CCN(C)CC2)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 5/20 0.42
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ACACB O00763 8/20 0.40
HRH4 Q9H3N8 1/20 0.39
KDM4E B2RXH2 1/20 0.38
PHGDH O43175 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
GFER P55789 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29676228 0.86 MAPK1 (0.42) MAPK1NPC1LMNATP53RAB9A
SCHEMBL17470867 0.78 ALDH1A1 (0.42) MAPK1NPC1LMNATP53RAB9A
SCHEMBL20738607 0.77 MAPK1 (0.44) MAPK1NPC1LMNATP53RAB9A
SCHEMBL18793895 0.77 MAPK1 (0.45) MAPK1NPC1LMNATP53RAB9A
SCHEMBL18794259 0.76 HRH4 (0.43) MAPK1NPC1LMNATP53RAB9A
SCHEMBL29675772 0.75 MAPK1 (0.59) MAPK1LMNA
SCHEMBL29338319 0.75 MAPK1 (0.46) MAPK1NPC1LMNATP53RAB9A
SCHEMBL29675508 0.75 MAPK1 (0.41) MAPK1LMNAACACBGFER
SCHEMBL23343854 0.74 MAPK1 (0.40) MAPK1NPC1LMNATP53RAB9A
SCHEMBL8259537 0.73 SMN1; SMN2 (0.53) NPC1LMNATP53RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108617166-B Protein kinase inhibitor benzolactam compounds 大冢制药株式会社 2022-05-17 CN claimed