SCHEMBL29675755

SCHEMBL29675755

CCC(=O)N[C@H](CO)c1ccnc(NC)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
ROCK2 O75116 3/20 0.37
MAPK1 P28482 3/20 0.36
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 1/20 0.36
RIPK1 Q13546 1/20 0.35
TYK2 P29597 2/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
ALOX12 P18054 4/20 0.35
ROCK1 Q13464 2/20 0.34
CYP3A4 P08684 1/20 0.34
RPS6KA5 O75582 1/20 0.34
MAP4K4 O95819 1/20 0.34
PRKACA P17612 1/20 0.34
RPS6KB1 P23443 1/20 0.34
AKT1 P31749 1/20 0.34
AKT2 P31751 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29675753 0.83 NPC1 (0.47) L3MBTL1NPC1RAB9AROCK2KDM4E
SCHEMBL29675931 0.80 MAPK1 (0.41) L3MBTL1NPC1RAB9AROCK2MAPK1
SCHEMBL20738649 0.80 KCNB1 (0.45) NPC1RAB9AROCK2MAPK1ROCK1
SCHEMBL29676371 0.76 CTSA (0.44) NPC1RAB9AMAPK1KDM4EALDH1A1
SCHEMBL29675688 0.74 MAPK1 (0.46) NPC1RAB9AROCK2MAPK1GSK3B
SCHEMBL29675681 0.74 ROCK2 (0.34) L3MBTL1NPC1RAB9AROCK2MAPK1
SCHEMBL29676029 0.73 PIK3CA (0.50) RAB9AMAPK1KDM4EGSK3B
SCHEMBL29675928 0.72 KCNH2 (0.40) L3MBTL1NPC1RAB9AMAPK1ALDH1A1
SCHEMBL18765697 0.71 CYP26A1 (0.47) ROCK2MAPK1KDM4EALDH1A1RIPK1
SCHEMBL31037006 0.71 MAPK1 (0.46) MAPK1ALDH1A1RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108617166-B Protein kinase inhibitor benzolactam compounds 大冢制药株式会社 2022-05-17 CN claimed