SCHEMBL29680755

SCHEMBL29680755

CCC(CCNCc1ccc(-c2nc(-c3ccccc3)c3ccn(-c4ccc(CNCCC(CC)N(C)C)cc4)c3n2)cc1)N(C)C

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
CDK1 P06493 1/20 0.33
SRC P12931 1/20 0.33
CSK P41240 1/20 0.33
ABL2 P42684 1/20 0.33
PDE4B Q07343 1/20 0.32
HDAC1 Q13547 1/20 0.31
USP2 O75604 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
TDP2 O95551 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29680480 0.97 TDP2 (0.32) PDE4BUSP2LMNACYP1A2CYP3A4
Oxalic Acid SCHEMBL29680919 0.96 KDM4E (0.35) ABL1EGFRCDK1SRCCSK
Oxalic Acid SCHEMBL29680387 0.93 KDM4E (0.37) PDE4BHDAC1USP2LMNACYP1A2
SCHEMBL29680662 0.89 HDAC1 (0.33) ABL1EGFRCDK1SRCCSK
SCHEMBL29680525 0.88 ENPP1 (0.32) HDAC1TDP2
SCHEMBL29680538 0.86 LSS (0.32) ABL1EGFRCDK1SRCCSK
Oxalic Acid SCHEMBL29680298 0.85 HDAC1 (0.36) ABL1EGFRCDK1SRCCSK
Oxalic Acid SCHEMBL29680467 0.85 KDM4E (0.36) PDE4BHDAC1USP2LMNACYP1A2
SCHEMBL29680879 0.83 TDP2 (0.32) PDE4BHDAC1LMNATDP2
SCHEMBL29680410 0.82 ALDH1A1 (0.42) ABL1EGFRCDK1SRCCSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP claimed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO claimed
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP disclosed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed