SCHEMBL29680662

SCHEMBL29680662

CC(CCNCc1ccc(-c2nc(-c3ccccc3)c3ccn(-c4ccc(CNCCC(C)N(C)C)cc4)c3n2)cc1)N(C)C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.33
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
CDK1 P06493 1/20 0.33
SRC P12931 1/20 0.33
CSK P41240 1/20 0.33
ABL2 P42684 1/20 0.33
PDE4B Q07343 2/20 0.33
CYP1A2 P05177 2/20 0.32
CYP2D6 P10635 2/20 0.32
ALDH1A1 P00352 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
USP2 O75604 1/20 0.32
LMNA P02545 1/20 0.32
CYP3A4 P08684 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
MGLL Q99685 1/20 0.31
MEN1 O00255 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29680538 0.97 LSS (0.32) HDAC1ABL1EGFRCDK1SRC
Oxalic Acid SCHEMBL29680298 0.96 HDAC1 (0.36) HDAC1ABL1EGFRCDK1SRC
Oxalic Acid SCHEMBL29680606 0.93 KDM4E (0.36) HDAC1PDE4BCYP1A2CYP2D6ALDH1A1
SCHEMBL29680865 0.90 MAPK1 (0.41) CDK1PDE4BALDH1A1LMNAMEN1
SCHEMBL29680755 0.89 ABL1 (0.33) HDAC1ABL1EGFRCDK1SRC
SCHEMBL29680879 0.88 TDP2 (0.32) HDAC1PDE4BALDH1A1LMNAMAPT
Oxalic Acid SCHEMBL29680212 0.87 ALDH1A1 (0.39) HDAC1CDK1PDE4BALDH1A1LMNA
SCHEMBL29680480 0.86 TDP2 (0.32) PDE4BCYP1A2CYP2D6ALDH1A1USP2
Oxalic Acid SCHEMBL29680919 0.85 KDM4E (0.35) HDAC1ABL1EGFRCDK1SRC
SCHEMBL29680410 0.83 ALDH1A1 (0.42) HDAC1ABL1EGFRCDK1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP claimed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO claimed
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP disclosed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed