SCHEMBL29682017

SCHEMBL29682017

Brc1ccc(C(Br)Br)c(C(Br)Br)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.37
AHR P35869 3/20 0.35
ALOX15 P16050 1/20 0.35
NR4A2 P43354 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HSP90AA1 P07900 1/20 0.33
TLR9 Q9NR96 1/20 0.33
S100A4 P26447 1/20 0.33
PTPRC P08575 1/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
METAP2 P50579 3/20 0.32
DYRK1A Q13627 2/20 0.32
NOS1 P29475 2/20 0.32
JAK2 O60674 2/20 0.32
BCL2 P10415 1/20 0.32
MCL1 Q07820 1/20 0.32
CHEK1 O14757 1/20 0.32
AURKA O14965 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1304745 1.00 CYP2A6 (0.37) CYP2A6AHRALOX15NR4A2ALDH1A1
SCHEMBL1539492 0.81 HSP90AA1 (0.42) CYP2A6AHRALOX15NR4A2ALDH1A1
SCHEMBL1569950 0.77 MAPK1 (0.36) CYP2A6AHRNR4A2ALDH1A1MAPK1
SCHEMBL15056090 0.77 DGAT1 (0.36) CYP2A6AHRALOX15NR4A2ALDH1A1
SCHEMBL3872105 0.77 APLNR (0.44) CYP2A6AHRNR4A2ALDH1A1KMT2A
SCHEMBL24416900 0.77 MAOB (0.39) CYP2A6AHRNR4A2ALDH1A1MAPK1
SCHEMBL1539565 0.74 GPR84 (0.33) ALDH1A1
SCHEMBL1683312 0.74 GPR84 (0.33) CSNK2A1GABRA1GABRB1
SCHEMBL396064 0.74 MAOB (0.44) CYP2A6AHRNR4A2NOS1MCL1
SCHEMBL2061830 0.72 GAA (0.41) ALOX15ALDH1A1MAPK1TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4448504-A1 NAPHTHALENE AND QUINOLINE ANALOGS AS RXFP1 AGONISTS Bristol-Myers Squibb Company (US) 2024-10-23 EP disclosed
CN-118414330-A Naphthalene and quinoline analogs as RXFP1 agonists 百时美施贵宝公司 2024-07-30 CN disclosed
WO-2023114818-A1 NAPHTHALENE AND QUINOLINE ANALOGS AS RXFP1 AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-06-22 WO disclosed
CN-114560885-B Sound-sensitive agent with low phototoxicity and preparation method and application thereof 北京理工大学 2023-03-14 CN disclosed
CN-114560885-A Sound-sensitive agent with low phototoxicity and preparation method and application thereof 北京理工大学 2022-05-31 CN disclosed