SCHEMBL2969916

SCHEMBL2969916

Cc1cccc(S)c1C#N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
CYP2C19 P33261 1/20 0.50
TSHR P16473 2/20 0.43
KDM4E B2RXH2 4/20 0.37
RECQL P46063 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
LMNA P02545 2/20 0.35
CYP2A6 P11509 1/20 0.35
ALDH1A1 P00352 4/20 0.34
MAPT P10636 1/20 0.34
PSMD14 O00487 1/20 0.34
COPS5 Q92905 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
UPP1 Q16831 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31010144 1.00 CYP1A2 (0.50) CYP1A2CYP2C19TSHRKDM4ERECQL
SCHEMBL102473 0.83 CYP1A2 (0.59) CYP1A2CYP2C19TSHRKDM4ELMNA
Ethane SCHEMBL2154002 0.80 CYP1A2 (0.57) CYP1A2CYP2C19TSHRKDM4ELMNA
SCHEMBL28349620 0.80 CYP1A2 (0.57) CYP1A2CYP2C19TSHRKDM4ELMNA
SCHEMBL30485186 0.74 TSHR (0.62) CYP1A2CYP2C19TSHRKDM4ETDP1
SCHEMBL3074213 0.74 MAOA (0.45) TSHRKDM4EALDH1A1MAPTMAOA
SCHEMBL1003690 0.74 TSHR (0.62) CYP1A2CYP2C19TSHRKDM4ETDP1
SCHEMBL17796263 0.74 CYP1A2 (0.52) CYP1A2CYP2C19TSHRKDM4ERECQL
SCHEMBL3860200 0.74 CYP1A2 (0.47) CYP1A2CYP2C19TSHRKDM4ELMNA
SCHEMBL103444 0.73 CYP1A2 (0.50) CYP1A2CYP2C19TSHRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024151638-A2 COMPOUNDS FOR FGFRS INHIBITORS COGENT BIOSCIENCES, INC. (US) 2024-07-18 WO disclosed
EP-3814331-B9 NOVEL LXR MODULATORS WITH BICYCLIC CORE MOIETY ORSOBIO INC (US) 2023-08-09 EP disclosed
US-20190211033-A1 ARYL, HETEROARYL, AND HETEROCYCLIC COMPOUNDS FOR TREATMENT OF MEDICAL DISORDERS ACHILLION PHARMACEUTICALS, INC. (US) 2019-07-11 US disclosed
CN-103347880-A Isoxazoline derivatives for controlling invertebrate pests NOVARTIS AG 2013-10-09 CN disclosed
US-7776847-B2 Benzisothiazoles useful for treating or preventing HCV infection RIGEL PHARMACEUTICALS, INC. (US) 2010-08-17 US disclosed
US-7776847-B2 Benzisothiazoles useful for treating or preventing HCV infection RIGEL PHARMACEUTICALS, INC. (US) 2010-08-17 US disclosed
US-7776847-B2 Benzisothiazoles useful for treating or preventing HCV infection RIGEL PHARMACEUTICALS, INC. (US) 2010-08-17 US disclosed
EP-1853573-A1 BENZISOTHIAZOLES USEFUL FOR TREATING OR PREVENTING HCV INFECTION Rigel Pharmaceuticals, Inc. (US) 2007-11-14 EP disclosed
US-20060229294-A1 Benzisothiazoles useful for treating or preventing HCV infection RIGEL PHARMACEUTICALS, INC. (US) 2006-10-12 US disclosed
WO-2006091858-A1 BENZISOTHIAZOLES USEFUL FOR TREATING OR PREVENTING HCV INFECTION RIGEL PHARMACEUTICALS, INC. (US) 2006-08-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190211033-A1 ARYL, HETEROARYL, AND HETEROCYCLIC COMPOUNDS FOR TREATMENT OF MEDICAL DISORDERS CFD, F12, F3 CYP1A2 94/4885CYP2C19 68/4885TSHR 744/4885
US-20060229294-A1 Benzisothiazoles useful for treating or preventing HCV infection HAVCR2, ZC3HAV1, MAVS CYP1A2 862/4885CYP2C19 1287/4885TSHR 4487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.