SCHEMBL29699221

SCHEMBL29699221

Cc1ccc(C)n1-c1cc(C(F)(F)F)c(C(F)(F)F)nc1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MYC P01106 13/20 0.44
ESR1 P03372 1/20 0.40
ALOX15 P16050 1/20 0.40
PTPN7 P35236 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PTPN1 P18031 1/20 0.39
GRIA1 P42261 1/20 0.39
GRIA2 P42262 1/20 0.39
GRIA3 P42263 1/20 0.39
GRIA4 P48058 1/20 0.39
NR4A1 P22736 3/20 0.39
CFTR P13569 2/20 0.38
NOTUM Q6P988 2/20 0.37
AXL P30530 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2372656 1.00 MYC (0.44) MYCESR1ALOX15PTPN7HSD17B10
SCHEMBL2372372 0.85 MYC (0.43) MYCHSD17B10CFTRNOTUMCNR1
SCHEMBL29699241 0.85 CFTR (0.45) MYCESR1ALOX15PTPN7HSD17B10
SCHEMBL2372056 0.85 CFTR (0.45) MYCESR1ALOX15PTPN7HSD17B10
SCHEMBL2373031 0.83 MYC (0.44) MYCESR1ALOX15PTPN7HSD17B10
SCHEMBL2372906 0.80 CFTR (0.44) MYCESR1ALOX15PTPN7HSD17B10
SCHEMBL2371674 0.80 RBP4 (0.39) MYCESR1ALOX15PTPN7HSD17B10
SCHEMBL2371716 0.79 CFTR (0.65) CFTR
SCHEMBL2372480 0.78 CFTR (0.40) MYCESR1ALOX15PTPN7HSD17B10
SCHEMBL13518970 0.78 CFTR (0.42) MYCHSD17B10NR4A1CFTRNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3980121-A1 PYRIDINE AND PYRAZINE DERIVATIVE FOR THE TREATMENT OF CF, COPD, AND BRONCHIECTASIS Novartis AG (CH) 2022-04-13 EP disclosed