SCHEMBL29699382

SCHEMBL29699382

CN1CCN[C@H](CNC(=O)c2nc(Br)c(C(F)(F)F)nc2N)C1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 5/20 0.36
HDAC4 P56524 2/20 0.35
CFTR P13569 11/20 0.35
HDAC6 Q9UBN7 1/20 0.35
PRKCB P05771 1/20 0.32
PRKCA P17252 1/20 0.32
FLT3 P36888 1/20 0.32
PRKCE Q02156 1/20 0.32
PRKCQ Q04759 1/20 0.32
PRKCD Q05655 1/20 0.32
ACVR1 Q04771 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2372852 1.00 ADRB1 (0.36) ADRB1HDAC4CFTRHDAC6PRKCB
SCHEMBL2372856 1.00 ADRB1 (0.36) ADRB1HDAC4CFTRHDAC6PRKCB
SCHEMBL29699237 0.73 DRD2 (0.46)
SCHEMBL2372239 0.73 DRD2 (0.46)
SCHEMBL2372244 0.73 DRD2 (0.46)
SCHEMBL4828955 0.72 ADRB1 (0.38) ADRB1
SCHEMBL4828950 0.72 ADRB1 (0.38) ADRB1
SCHEMBL14784270 0.70 CFTR (0.42) CFTR
SCHEMBL2373230 0.70 HDAC4 (0.41) HDAC4HDAC6
SCHEMBL29699276 0.70 CD274 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3980121-A1 PYRIDINE AND PYRAZINE DERIVATIVE FOR THE TREATMENT OF CF, COPD, AND BRONCHIECTASIS Novartis AG (CH) 2022-04-13 EP disclosed