SCHEMBL29707102

SCHEMBL29707102

COC(=O)c1cc(-c2cc(F)c(OC)cc2F)ncc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 2/20 0.43
JMJD6 Q6NYC1 1/20 0.40
TGFBR1 P36897 2/20 0.39
KDM4E B2RXH2 4/20 0.38
AAK1 Q2M2I8 1/20 0.37
CTSA P10619 2/20 0.36
DHODH Q02127 2/20 0.36
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
POLB P06746 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
ACVR1B P36896 1/20 0.35
ACVRL1 P37023 1/20 0.35
GAA P10253 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22981650 1.00 ALPL (0.43) ALPLJMJD6TGFBR1KDM4EAAK1
SCHEMBL22981788 0.89 ALPL (0.54) ALPLJMJD6TGFBR1KDM4EDHODH
SCHEMBL22986367 0.82 CDK9 (0.46) ALPLJMJD6ROCK2ROCK1SLC6A4
SCHEMBL29707061 0.80 DHODH (0.47) JMJD6KDM4EDHODHROCK2GAA
SCHEMBL22981957 0.80 DHODH (0.47) JMJD6KDM4EDHODHROCK2GAA
SCHEMBL22986361 0.78 JMJD6 (0.44) ALPLJMJD6TGFBR1KDM4EDHODH
SCHEMBL17700427 0.77 KDM4E (0.50) KDM4EPOLBGAA
SCHEMBL22986360 0.77 TGFBR1 (0.41) ALPLJMJD6TGFBR1KDM4EAAK1
SCHEMBL22986364 0.75 JMJD6 (0.41) JMJD6KDM4EDHODHPOLBSLC6A4
SCHEMBL22986363 0.74 KDM4E (0.49) ALPLJMJD6TGFBR1KDM4EDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114585622-B Piperidinyl-methyl-purinamines as NSD2 inhibitors and anticancer agents 诺华股份有限公司 2024-08-09 CN disclosed
CN-114585622-A Piperidinyl-methyl-purinamines as NSD2 inhibitors and anticancer agents 诺华股份有限公司 2022-06-03 CN disclosed