SCHEMBL29707609

SCHEMBL29707609

CC(C)(C)c1ccc(Nc2cncc(Br)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 2/20 0.49
XDH P47989 1/20 0.49
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
NAMPT P43490 1/20 0.38
SLC2A1 P11166 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
HTT P42858 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
FGFR2 P21802 1/20 0.36
DHODH Q02127 1/20 0.35
CSNK1A1 P48729 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28824305 1.00 SLC22A12 (0.49) SLC22A12XDHCYP1A2CYP3A4CYP2C9
SCHEMBL28824302 0.81 CHRNB4 (0.48) SLC22A12XDHCYP1A2CYP3A4CYP2C19
SCHEMBL28801068 0.78 RAPGEF4 (0.44) NPC1RAB9ASMN1; SMN2POLBHTT
SCHEMBL30494419 0.77 CHRNB4 (0.48) SLC22A12XDHRAB9ACHRNB4CHRNA3
SCHEMBL26465213 0.77 CHRNB4 (0.48) SLC22A12XDHRAB9ACHRNB4CHRNA3
SCHEMBL4156639 0.77 SCN9A (0.54) SLC22A12XDHCHRNB4CHRNA3ALDH1A1
SCHEMBL29707607 0.77 SCN9A (0.54) SLC22A12XDHCHRNB4CHRNA3ALDH1A1
SCHEMBL4147660 0.77 HSD17B10 (0.48) SLC22A12XDHCYP3A4CHRNB4CHRNA3
SCHEMBL2821463 0.77 RAB9A (0.57) SLC22A12XDHNPC1RAB9ACHRNB4
SCHEMBL2392625 0.75 TSHR (0.52) NPC1RAB9ASMN1; SMN2ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114805192-B Tricyclic XOR/URAT1 dual inhibitor containing 2-hydroxybenzoic acid and preparation method and application thereof 华南理工大学 2023-05-23 CN disclosed
CN-114805192-A Tricyclic XOR/URAT1 dual inhibitor containing 2-hydroxybenzoic acid and preparation method and application thereof 华南理工大学 2022-07-29 CN disclosed