SCHEMBL29709653

SCHEMBL29709653

Cc1c(B2OC(C)(C)C(C)(C)O2)cccc1N(C)C(=O)c1nccs1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BTK Q06187 4/20 0.40
GRM4 Q14833 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HSD17B1 P14061 1/20 0.33
HSD17B2 P37059 1/20 0.33
PLA2G7 Q13093 1/20 0.32
JAK2 O60674 3/20 0.31
LPL P06858 1/20 0.31
LIPG Q9Y5X9 1/20 0.31
NR3C1 P04150 1/20 0.31
KMT2A Q03164 1/20 0.31
RBBP9 O75884 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16336718 1.00 BTK (0.40) BTKGRM4ALDH1A1HSD17B1HSD17B2
SCHEMBL16337053 0.77 BTK (0.43) BTKGRM4
SCHEMBL29709486 0.77 BTK (0.43) BTKGRM4
SCHEMBL17699662 0.73 BTK (0.40) BTKJAK2
SCHEMBL29782721 0.73 BTK (0.40) BTKJAK2
SCHEMBL18976231 0.69 JAK2 (0.37) BTKHSD17B1HSD17B2JAK2
SCHEMBL16320402 0.69 POLB (0.40) ALDH1A1KMT2A
SCHEMBL18985009 0.66 JAK2 (0.35) BTKALDH1A1JAK2LPLLIPG
SCHEMBL11927624 0.66 LPL (0.44) BTKJAK2LPLLIPG
SCHEMBL16336876 0.66 GRM4 (0.45) BTKGRM4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4008328-A1 PRIMARY CARBOXAMIDES AS BTK INHIBITORS AbbVie Inc. (US) 2022-06-08 EP disclosed