SCHEMBL2970978

SCHEMBL2970978

FC(F)(F)c1cccc2c1[CH]c1ccccc1-2

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.39
HSD11B1 P28845 4/20 0.38
CES1 P23141 1/20 0.37
NOTUM Q6P988 1/20 0.36
GPR3 P46089 1/20 0.35
ALDH1A1 P00352 3/20 0.35
CYP1A2 P05177 3/20 0.35
CYP2C19 P33261 3/20 0.35
CYP3A4 P08684 1/20 0.35
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KIF11 P52732 1/20 0.34
HPGD P15428 1/20 0.34
AR P10275 1/20 0.34
SCN9A Q15858 1/20 0.34
PSMB8 P28062 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2964849 0.90 HSD11B1 (0.41) PDK2HSD11B1CES1NOTUMALDH1A1
SCHEMBL18242471 0.85 PDK2 (0.30) PDK2
SCHEMBL18241988 0.82
SCHEMBL18242355 0.80
SCHEMBL2975651 0.80 HSD11B1 (0.37) PDK2HSD11B1NOTUMALDH1A1CYP1A2
SCHEMBL5597066 0.80 CA2 (0.31) ALDH1A1TDP1
SCHEMBL18242204 0.80 TSHR (0.30)
SCHEMBL726454 0.80 CA2 (0.40) ALDH1A1TDP1KIF11
SCHEMBL2963747 0.79 HSD11B1 (0.36) HSD11B1NOTUMGPR3ALDH1A1CYP1A2
SCHEMBL18244028 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611131-B1 PYRAZOLOPYRIDINE DERIVATES PALAU PHARMA SA (ES) 2010-09-15 EP claimed