SCHEMBL29746469

SCHEMBL29746469

Clc1ccc2c(Cl)cccc2n1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.46
CYP2A6 P11509 2/20 0.46
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
GUSB P08236 1/20 0.40
BACE1 P56817 1/20 0.39
P2RX7 Q99572 3/20 0.39
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
NR4A2 P43354 1/20 0.37
TYMS P04818 2/20 0.37
BCHE P06276 1/20 0.37
C1R P00736 1/20 0.37
NOS1 P29475 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL239860 1.00 CYP1A2 (0.46) CYP1A2CYP2A6MAOAMAOBPDE3B
SCHEMBL3071480 0.83 BACE1 (0.60) CYP1A2CYP2A6BACE1NR4A2TYMS
SCHEMBL13077349 0.80 MAOA (0.41) CYP1A2MAOAMAOBCYP3A4TSHR
SCHEMBL1615737 0.78 ACHE (0.45) CYP1A2MAOAMAOBTSHRBACE1
SCHEMBL116741 0.78 ALDH1A1 (0.50) CYP1A2MAOAMAOBCYP3A4TSHR
SCHEMBL7219172 0.78 CYP1A2 (0.44) CYP1A2CYP2A6MAOAMAOBPDE3B
SCHEMBL707745 0.78 BACE1 (0.66) CYP1A2MAOAMAOBCYP3A4TSHR
SCHEMBL7045373 0.78 CYP1A2 (0.42) CYP1A2CYP2A6MAOAMAOBPDE3B
SCHEMBL29980068 0.78 CYP1A2 (0.42) CYP1A2CYP2A6MAOAMAOBPDE3B
SCHEMBL3338347 0.78 MAOA (0.40) MAOAMAOBCYP3A4TSHRBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116348112-A Imidazopiperazine inhibitors of transcriptional activator proteins 德州大学系统董事会 2023-06-27 CN disclosed
WO-2022138888-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF 東レ株式会社 2022-06-30 WO disclosed