SCHEMBL29756331

SCHEMBL29756331

COc1ccc(-c2cc(Cl)cc3c4ccnc(C)c4n(C)c23)cc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 13/20 0.55
MAOA P21397 2/20 0.55
ACHE P22303 2/20 0.55
BCHE P06276 1/20 0.55
HASPIN Q8TF76 6/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
DYRK2 Q92630 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20122972 1.00 DYRK1A (0.55) DYRK1AMAOAACHEBCHEHASPIN
SCHEMBL20123007 0.85 DYRK1A (0.58) DYRK1AMAOAACHEBCHEHASPIN
SCHEMBL30664315 0.85 DYRK1A (0.58) DYRK1AMAOAACHEBCHEHASPIN
SCHEMBL20122960 0.81 DYRK1A (0.45) DYRK1AMAOAACHEBCHEHASPIN
SCHEMBL30664227 0.81 DYRK1A (0.45) DYRK1AMAOAACHEBCHEHASPIN
SCHEMBL20122936 0.79 AURKA (0.41) DYRK1AMAOAACHEBCHE
SCHEMBL20123059 0.78 HASPIN (0.43) DYRK1AMAOAACHEBCHEHASPIN
SCHEMBL30664168 0.78 HASPIN (0.43) DYRK1AMAOAACHEBCHEHASPIN
SCHEMBL20122851 0.76 DYRK1A (0.47) DYRK1AMAOAACHEBCHEHASPIN
SCHEMBL28654194 0.75 ACHE (0.80) DYRK1AMAOAACHEBCHEHASPIN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110382496-B Substituted pyrido [3,4-b ] indoles for the treatment of cartilage disorders 赛诺菲 2022-08-09 CN claimed
US-20250333412-A1 SUBSTITUTED PYRIDO[3,4-B]INDOLES FOR THE TREATMENT OF CARTILAGE DISORDERS SANOFI SA (FR) 2025-10-30 US disclosed
CN-110382496-B Substituted pyrido [3,4-b ] indoles for the treatment of cartilage disorders 赛诺菲 2022-08-09 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250333412-A1 SUBSTITUTED PYRIDO[3,4-B]INDOLES FOR THE TREATMENT OF CARTILAGE DISORDERS COL2A1, IDO1, COL1A1 DYRK1A 498/4885MAOA 246/4885ACHE 2583/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.