SCHEMBL29763523

SCHEMBL29763523

COc1nccc(CF)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 7/20 0.38
GRIN2B Q13224 7/20 0.38
NOS3 P29474 2/20 0.37
NOS1 P29475 2/20 0.37
NOS2 P35228 2/20 0.37
CCR1 P32246 1/20 0.36
CCR5 P51681 1/20 0.36
CCR8 P51685 1/20 0.36
FFAR1 O14842 1/20 0.35
PDPK1 O15530 1/20 0.34
RAB9A P51151 1/20 0.33
RXRA P19793 5/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18200291 0.82 NOS3 (0.38) GRIN1GRIN2BNOS3NOS1NOS2
SCHEMBL16815694 0.80 CCR1 (0.39) GRIN1GRIN2BNOS3NOS1NOS2
SCHEMBL1154350 0.80 LOXL2 (0.43) GRIN1GRIN2BNOS3NOS1NOS2
SCHEMBL20893799 0.80 GRIN1 (0.38) GRIN1GRIN2BNOS3NOS1NOS2
SCHEMBL19932063 0.80 NOS3 (0.37) GRIN1GRIN2BNOS3NOS1NOS2
SCHEMBL30026942 0.79 GRIN1 (0.36) GRIN1GRIN2BNOS3NOS1NOS2
SCHEMBL22905296 0.77 FFAR1 (0.36) GRIN1GRIN2BNOS3NOS1NOS2
SCHEMBL21567109 0.77 GRIN1 (0.36) GRIN1GRIN2BNOS3NOS1NOS2
SCHEMBL990352 0.77 KCNH2 (0.52) NOS3NOS1NOS2FFAR1ALDH1A1
SCHEMBL5103633 0.76 MEN1 (0.39) GRIN1GRIN2BNOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4288424-A1 NOVEL HETEROARYL-SUBSTITUTED IMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2023-12-13 EP disclosed
WO-2022167631-A1 NOVEL HETEROARYL-SUBSTITUTED IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2022-08-11 WO disclosed