SCHEMBL29772902

SCHEMBL29772902

OCc1ccccc1N1CCN(c2ccc(Cl)cc2F)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.49
GRM2 Q14416 1/20 0.49
AKR1C3 P42330 1/20 0.49
GRM5 P41594 1/20 0.47
KMT2A Q03164 7/20 0.47
L3MBTL1 Q9Y468 2/20 0.45
MEN1 O00255 4/20 0.44
SLC6A2 P23975 1/20 0.43
SLC6A3 Q01959 1/20 0.43
MAPT P10636 5/20 0.43
MAPK1 P28482 3/20 0.43
ALDH1A1 P00352 3/20 0.43
LMNA P02545 3/20 0.43
PHGDH O43175 1/20 0.43
GAA P10253 2/20 0.42
CYP2C19 P33261 1/20 0.42
GFER P55789 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HTT P42858 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21261309 1.00 DRD4 (0.49) DRD4GRM2AKR1C3GRM5KMT2A
SCHEMBL23536030 0.81 GRM2 (0.43) GRM2AKR1C3KMT2A
SCHEMBL4960474 0.80 KDM4E (0.52) DRD4AKR1C3SLC6A2SLC6A3ALDH1A1
SCHEMBL21261239 0.79 POLB (0.54) DRD4GRM2GRM5KMT2AL3MBTL1
SCHEMBL21261308 0.79 TSHR (0.45) DRD4GRM2GRM5KMT2AL3MBTL1
SCHEMBL29772857 0.79 TSHR (0.45) DRD4GRM2GRM5KMT2AL3MBTL1
SCHEMBL30233081 0.78 HPGD (0.53) DRD4GRM2AKR1C3L3MBTL1MAPT
SCHEMBL21261310 0.78 MAPT (0.47) DRD4GRM2KMT2AL3MBTL1MEN1
SCHEMBL23535932 0.77 ENPP2 (0.53) DRD4GRM2GRM5KMT2AL3MBTL1
SCHEMBL21261350 0.76 SMN1; SMN2 (0.49) DRD4GRM2GRM5KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022150461-A1 MODULATORS OF TRPML, THEIR COMPOSITIONS AND METHODS OF USE CARAWAY THERAPEUTICS, INC. (US) 2022-07-14 WO disclosed