SCHEMBL29778012

SCHEMBL29778012

Cc1ccc(S(=O)(=O)n2c(C(c3ccccc3)P(=O)(c3cccs3)c3cccs3)c(-c3ccccc3)c3ccccc32)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PCSK9 Q8NBP7 3/20 0.44
AGTR1 P30556 3/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
HTR6 P50406 4/20 0.38
CYP19A1 P11511 1/20 0.38
NOD2 Q9HC29 2/20 0.36
NOD1 Q9Y239 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
KDM4E B2RXH2 1/20 0.35
UBE2N P61088 1/20 0.35
GBA1 P04062 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29778016 0.86 PCSK9 (0.48) PCSK9AGTR1L3MBTL1HTR6CYP19A1
SCHEMBL29778015 0.83 PCSK9 (0.44) PCSK9AGTR1L3MBTL1HTR6NOD2
SCHEMBL28400037 0.79 AGTR1 (0.41) PCSK9AGTR1L3MBTL1HTR6CYP19A1
SCHEMBL29778010 0.79 AGTR1 (0.41) PCSK9AGTR1L3MBTL1HTR6CYP19A1
SCHEMBL28402229 0.79 PCSK9 (0.44) PCSK9AGTR1L3MBTL1HTR6NOD1
SCHEMBL28397417 0.79 HTR6 (0.42) PCSK9AGTR1L3MBTL1HTR6CYP19A1
SCHEMBL28790159 0.78 PCSK9 (0.48) PCSK9AGTR1L3MBTL1HTR6NOD2
SCHEMBL28408113 0.76 PCSK9 (0.46) PCSK9AGTR1L3MBTL1HTR6NOD2
SCHEMBL29778014 0.76 PCSK9 (0.46) PCSK9AGTR1L3MBTL1HTR6NOD2
SCHEMBL28398527 0.75 AGTR1 (0.45) PCSK9AGTR1L3MBTL1HTR6CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111187298-B C2-phosphono methylene indole compound and preparation method and application thereof 成都大学 2022-07-19 CN disclosed