SCHEMBL29779476

SCHEMBL29779476

O=C([C@@H]1CCCN1c1ccc(Br)cc1)N1CCOCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.54
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
ROCK2 O75116 1/20 0.46
ROCK1 Q13464 1/20 0.46
CDC42BPB Q9Y5S2 1/20 0.46
PHGDH O43175 1/20 0.46
MGLL Q99685 1/20 0.45
GPR183 P32249 1/20 0.43
KCNH2 Q12809 1/20 0.43
POLB P06746 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16197772 0.79 SMN1; SMN2 (0.44) MEN1KMT2AALDH1A1HSD17B10RXFP1
SCHEMBL3060275 0.79 SMN1; SMN2 (0.44) MEN1KMT2AALDH1A1HSD17B10RXFP1
SCHEMBL3060271 0.79 SMN1; SMN2 (0.44) MEN1KMT2AALDH1A1HSD17B10RXFP1
SCHEMBL11985533 0.78 CNR2 (0.41) ALDH1A1RXFP1
SCHEMBL29779383 0.77 ALDH1A1 (0.51) AKR1C3MEN1KMT2AALDH1A1PHGDH
SCHEMBL22798963 0.75 BRS3 (0.44) MEN1KMT2AALDH1A1GPR183L3MBTL1
SCHEMBL3315348 0.74 ALDH1A1 (0.42) AKR1C3MEN1KMT2AALDH1A1TSHR
SCHEMBL3312862 0.72 ALDH1A1 (0.53) MEN1KMT2AALDH1A1POLBNPC1
SCHEMBL14711760 0.71 ALDH1A1 (0.48) MEN1KMT2AALDH1A1TSHRPOLB
SCHEMBL9367926 0.71 ADAM10 (0.44) KMT2AL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114716370-A Pyridine-containing polycyclic derivative inhibitor, and preparation method and application thereof 上海翰森生物医药科技有限公司 2022-07-08 CN disclosed