SCHEMBL29795308

SCHEMBL29795308

COc1ccc(CN(C(=O)OC(C)(C)C)C2CCN(C(=O)OC(C)(C)C)C2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.60
GPR119 Q8TDV5 3/20 0.53
ALDH1A1 P00352 1/20 0.51
JAK2 O60674 1/20 0.49
JAK1 P23458 1/20 0.49
NR1D1 P20393 1/20 0.47
USP30 Q70CQ3 2/20 0.47
STS P08842 1/20 0.47
HTR2A P28223 1/20 0.47
EPHX2 P34913 1/20 0.46
UBE2M P61081 1/20 0.46
DCUN1D1 Q96GG9 1/20 0.46
SLC2A1 P11166 1/20 0.45
TP53 P04637 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HTT P42858 1/20 0.44
OPRM1 P35372 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30954953 0.83 GPR119 (0.52) GPR119ALDH1A1JAK2JAK1NR1D1
SCHEMBL34474238 0.82 GPR119 (0.50) HSD11B1GPR119ALDH1A1JAK2JAK1
SCHEMBL4263388 0.81 GPR119 (0.54) HSD11B1GPR119ALDH1A1JAK2JAK1
SCHEMBL1624526 0.81 HSD11B1 (0.66) HSD11B1GPR119JAK2JAK1NR1D1
SCHEMBL24424613 0.81 GPR119 (0.49) GPR119ALDH1A1JAK2JAK1NR1D1
SCHEMBL30954995 0.80 GPR119 (0.48) HSD11B1GPR119ALDH1A1JAK2JAK1
SCHEMBL4212846 0.80 HTR2A (0.56) GPR119ALDH1A1STSHTR2AEPHX2
SCHEMBL4215215 0.79 GPR119 (0.52) GPR119ALDH1A1HTR2AEPHX2UBE2M
SCHEMBL25609126 0.79 HTR2A (0.46) HSD11B1ALDH1A1NR1D1HTR2AUBE2M
SCHEMBL19123612 0.79 ALDH1A1 (0.51) GPR119ALDH1A1JAK2JAK1NR1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114761412-A Substituted macrocyclic compounds and related methods of treatment 阿尔克姆斯有限公司 2022-07-15 CN disclosed