SCHEMBL29797145

SCHEMBL29797145

CCOC(=O)/C=C/c1nc(CCCc2ccc3c(n2)N(C(=O)OC(C)(C)C)CCC3)cs1

nearest known ligand 0.32

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
MPO P05164 1/20 0.32
HDAC3 O15379 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC7 Q8WUI4 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC10 Q969S8 1/20 0.30
HDAC11 Q96DB2 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
HDAC9 Q9UKV0 1/20 0.30
HDAC5 Q9UQL6 1/20 0.30
NCOR2 Q9Y618 1/20 0.30
ACKR3 P25106 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21311563 1.00 ALDH1A1 (0.32) ALDH1A1MPOHDAC3HDAC4HDAC1
SCHEMBL20141485 0.89 ALDH1A1 (0.36) ALDH1A1HDAC3HDAC4HDAC1HDAC7
SCHEMBL20141482 0.89 ALDH1A1 (0.36) ALDH1A1HDAC3HDAC4HDAC1HDAC7
SCHEMBL17921404 0.79 HPGD (0.37) ALDH1A1MPO
SCHEMBL29416368 0.79 HPGD (0.37) ALDH1A1MPO
SCHEMBL24908851 0.79 MPO (0.39) ALDH1A1MPO
SCHEMBL1840941 0.78 MPO (0.39) ALDH1A1MPO
SCHEMBL21314483 0.78 ITGAV (0.37) MPO
SCHEMBL22223283 0.78 KDM4E (0.36) ALDH1A1MPO
SCHEMBL16607378 0.78 KDM4E (0.36) ALDH1A1MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11884661-B2 3-substituted propionic acids as αV integrin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2024-01-30 US disclosed
EP-3538525-B1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-06-22 EP disclosed
CN-110167935-B 3-substituted propionic acids as alpha V integrin inhibitors 百时美施贵宝公司 2022-05-27 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11884661-B2 3-substituted propionic acids as αV integrin inhibitors ITGB3, ITGB1, ITGAV ALDH1A1 504/4885MPO 4599/4885HDAC3 231/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.