SCHEMBL29801

SCHEMBL29801

O=C(c1ccc(Oc2ccccc2)c(O)c1)c1nc2ccc(O)cc2s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 9/20 1.00
HSD17B2 P37059 9/20 1.00
CYP1A2 P05177 2/20 0.63
CYP3A4 P08684 2/20 0.63
CYP2D6 P10635 2/20 0.63
CYP2C9 P11712 2/20 0.63
CYP2B6 P20813 2/20 0.63
CYP2C19 P33261 2/20 0.63
TTR P02766 1/20 0.52
BCL2 P10415 1/20 0.51
MCL1 Q07820 1/20 0.51
BAD Q92934 1/20 0.51
MAOB P27338 7/20 0.47
MAPT P10636 1/20 0.46
SNCA P37840 1/20 0.46
PDE10A Q9Y233 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8401047 0.84 HSD17B1 (0.72) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL8400538 0.80 HSD17B1 (0.81) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL31420 0.78 HSD17B1 (0.64) HSD17B1HSD17B2TTRBCL2MCL1
SCHEMBL30049 0.78 HSD17B1 (0.76) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL29654 0.77 HSD17B1 (1.00) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL29673 0.77 HSD17B1 (1.00) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL8402863 0.77 HSD17B1 (0.68) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL8401031 0.77 HSD17B1 (0.74) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL29786 0.77 HSD17B1 (1.00) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL8401357 0.76 HSD17B1 (0.63) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed