SCHEMBL29802464

SCHEMBL29802464

CS(=O)(=O)c1ccc(-c2nc(Br)cnc2N)cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.56
ATR Q13535 10/20 0.49
PRKDC P78527 5/20 0.49
ATM Q13315 4/20 0.49
MAP4K4 O95819 3/20 0.48
MINK1 Q8N4C8 2/20 0.48
FYN P06241 2/20 0.48
TNIK Q9UKE5 1/20 0.48
PIK3CA P42336 1/20 0.46
PI4KB Q9UBF8 1/20 0.46
DHFR P00374 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23093419 1.00 KCNH2 (0.56) KCNH2ATRPRKDCATMMAP4K4
SCHEMBL23093414 0.83 KCNH2 (0.55) KCNH2ATRPRKDCATMMAP4K4
SCHEMBL23093139 0.81 LRRK2 (0.48) KCNH2ATRFYN
SCHEMBL16425220 0.80 KCNH2 (0.69) KCNH2ATRPRKDCATM
SCHEMBL23093191 0.79 PTGS2 (0.42)
SCHEMBL29802518 0.79 PTGS2 (0.42)
SCHEMBL20371190 0.78 ABL1 (0.46) ATRMAP4K4
SCHEMBL12488659 0.78 ALDH1A1 (0.41) ATRATM
SCHEMBL23093381 0.77 PTGS2 (0.43) KCNH2
SCHEMBL29802439 0.77 PTGS2 (0.43) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4027993-A1 CYCLOOXYGENASE-2 INHIBITORS AND USES THEREOF The Broad Institute Inc. (US) 2022-07-20 EP disclosed