SCHEMBL29804262

SCHEMBL29804262

CC(=O)OC(F)(F)F.CCOC(=O)c1cnco1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
NAMPT P43490 1/20 0.38
KDM4E B2RXH2 5/20 0.36
ALDH1A1 P00352 4/20 0.36
HPGD P15428 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
CDC7 O00311 1/20 0.34
DBF4 Q9UBU7 1/20 0.34
ACACB O00763 2/20 0.34
CYP1A2 P05177 1/20 0.34
MAPT P10636 2/20 0.33
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL414791 0.85 NAMPT (0.46) HDAC4HDAC6NAMPTALDH1A1CYP2C9
Hydrochloric Acid SCHEMBL29099329 0.84 NAMPT (0.45) HDAC4HDAC6NAMPTALDH1A1CYP2C9
SCHEMBL28317573 0.73 ALDH1A1 (0.44) NAMPTKDM4EALDH1A1SMN1; SMN2ACACB
SCHEMBL23042189 0.70 CHRNA4 (0.36) ALDH1A1SMN1; SMN2CYP2C9CYP2C19ACACB
SCHEMBL3139874 0.67 ALDH1A1 (0.35) NAMPTALDH1A1ACACBMAPTMEN1
SCHEMBL15419308 0.66 NPC1 (0.46) ALDH1A1ACACBCYP1A2MAPTHTT
SCHEMBL15465637 0.66 HDAC4 (0.40) HDAC4HDAC6NAMPTKDM4EALDH1A1
Hydrochloric Acid SCHEMBL28665424 0.66 CHRNA4 (0.41) KDM4EALDH1A1CYP2C19ACACBCYP1A2
SCHEMBL3827774 0.64 TBXAS1 (0.43) KDM4EALDH1A1HPGDSMN1; SMN2CYP2C19
SCHEMBL29088542 0.63 ALDH1A1 (0.41) KDM4EALDH1A1HPGDPOLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114874222-A Carrying non-aromatic P2 , Novel macrocyclic form of factor XIA 百时美施贵宝公司 2022-08-09 CN disclosed
CN-114805365-A Carrying non-aromatic P2 , Novel macrocyclic form of factor XIA 百时美施贵宝公司 2022-07-29 CN disclosed