SCHEMBL29809015

SCHEMBL29809015

C[C@H](N)c1ccc(F)c(C#N)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.42
ADRB1 P08588 2/20 0.42
PGR P06401 2/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
ADRB3 P13945 1/20 0.38
PIK3CD O00329 1/20 0.38
ABL1 P00519 1/20 0.38
EGFR P00533 1/20 0.38
HCK P08631 1/20 0.38
SRC P12931 1/20 0.38
KDR P35968 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
MTOR P42345 1/20 0.38
PIK3CG P48736 1/20 0.38
EPHB4 P54760 1/20 0.38
PRKDC P78527 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28802853 1.00 ADRB2 (0.42) ADRB2ADRB1PGRCYP1A2CYP3A4
SCHEMBL1240016 1.00 ADRB2 (0.42) ADRB2ADRB1PGRCYP1A2CYP3A4
Hydrochloric Acid SCHEMBL28802793 0.98 ADRB2 (0.41) ADRB2ADRB1PGRCYP1A2CYP3A4
Hydrochloric Acid SCHEMBL3703483 0.98 ADRB2 (0.41) ADRB2ADRB1PGRCYP1A2CYP3A4
SCHEMBL16649615 0.85 TRPV4 (0.48) ADRB2ADRB1PIK3CDABL1EGFR
SCHEMBL22495734 0.85 TRPV4 (0.48) ADRB2ADRB1PIK3CDABL1EGFR
SCHEMBL28802774 0.85 TRPV4 (0.48) ADRB2ADRB1PIK3CDABL1EGFR
SCHEMBL879123 0.85 PGR (0.43) ADRB2ADRB1PGRCYP1A2CYP3A4
Hydrochloric Acid SCHEMBL28803022 0.84 TRPV4 (0.47) ADRB2ADRB1PIK3CDABL1EGFR
SCHEMBL30892077 0.82 CYP11B1 (0.45) ADRB2ADRB1PGRCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114835687-B AhR inhibitors 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-114835687-A AhR inhibitors 重庆华森制药股份有限公司 2022-08-02 CN disclosed