SCHEMBL29824345

SCHEMBL29824345

Nc1nc2cnc(NC3CCCC3)nc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 1/20 0.47
ABL1 P00519 1/20 0.46
RIN1 Q13671 1/20 0.46
ULK1 O75385 1/20 0.44
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
MAPK8 P45983 4/20 0.41
HPGDS O60760 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
CDK4 P11802 3/20 0.39
CCND1 P24385 3/20 0.39
CDK1 P06493 2/20 0.39
CCNB1 P14635 2/20 0.39
CCNA2 P20248 2/20 0.39
CDK2 P24941 2/20 0.39
CCNA1 P78396 2/20 0.39
CTSK P43235 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7662487 0.75 PAK1 (0.60) PAK1ULK1KDM4EGAAMAPK8
SCHEMBL15264144 0.74 PAK1 (0.62) PAK1ULK1KDM4EGAAMAPK8
SCHEMBL9704728 0.73 PDE4A (0.43) PAK1ULK1KDM4EGAACDK4
SCHEMBL1551868 0.72 PAK1 (0.56) PAK1ULK1KDM4EGAAMAPK8
SCHEMBL14391351 0.71 MAPK8 (0.60) PAK1MAPK8MAPK9MAPK10MAPK14
SCHEMBL11000513 0.70 PAK1 (0.47) PAK1ULK1KDM4EGAAMAPK8
SCHEMBL22278819 0.69 ULK1 (0.41) PAK1ULK1MAPK8TYRO3EGFR
SCHEMBL1644969 0.69 ALDH1A1 (0.38) KDM4E
SCHEMBL10999501 0.69 PAK1 (0.49) PAK1ULK1KDM4EGAAMAPK8
SCHEMBL10998140 0.69 PAK1 (0.49) PAK1ULK1KDM4EGAAMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3464287-B1 ANIMAL AND HUMAN ANTI-MALARIAL AGENTS CELGENE CORP (US) 2022-06-08 EP claimed