SCHEMBL9704728

SCHEMBL9704728

CCCCc1nc2cnc(NC3CCCCC3)nc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
PAK1 Q13153 1/20 0.42
CDK4 P11802 2/20 0.41
CCND1 P24385 2/20 0.41
CCND2 P30279 1/20 0.41
CCND3 P30281 1/20 0.41
FLT3 P36888 7/20 0.41
TYRO3 Q06418 7/20 0.41
MERTK Q12866 7/20 0.41
GAS6 Q14393 7/20 0.41
LMNA P02545 1/20 0.40
AXL P30530 1/20 0.40
ULK1 O75385 1/20 0.38
ADORA3 P0DMS8 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNA2 P20248 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9704732 0.82 PAK1 (0.53) PDE4APDE4BPDE4CPDE4DPAK1
SCHEMBL9704929 0.77 PARP1 (0.40) FLT3TYRO3MERTKGAS6AXL
SCHEMBL29824345 0.73 PAK1 (0.47) PAK1CDK4CCND1CCND2CCND3
SCHEMBL9669702 0.72 PARP1 (0.42) TYRO3
SCHEMBL9705991 0.72 PARP1 (0.47) PDE4APDE4BPDE4CPDE4DLMNA
SCHEMBL9706003 0.70 PARP1 (0.40)
SCHEMBL9705258 0.70 PARP1 (0.40) CDK1CCNB1CDK2
SCHEMBL15264144 0.69 PAK1 (0.62) PAK1CDK4CCND1FLT3TYRO3
SCHEMBL7662487 0.67 PAK1 (0.60) PAK1CDK4CCND1FLT3TYRO3
SCHEMBL7851162 0.67 PARP1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470543-A1 Heterocyclic imidazoles, remedies containing them and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-02-12 EP disclosed