SCHEMBL29856430

SCHEMBL29856430

CN1CCN(Cc2ccc(NC(=O)c3ccccc3)cc2F)CC1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRAF P15056 4/20 0.62
KIT P10721 6/20 0.58
BTK Q06187 1/20 0.55
RAB9A P51151 3/20 0.54
NPC1 O15118 2/20 0.54
MAPT P10636 2/20 0.54
LMNA P02545 1/20 0.54
ABL1 P00519 1/20 0.51
LYN P07948 1/20 0.51
BCR P11274 1/20 0.51
EGFR P00533 2/20 0.50
RET P07949 2/20 0.50
FGFR1 P11362 1/20 0.50
KDR P35968 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29856263 0.90 KIT (0.61) BRAFKITBTKRAB9ANPC1
SCHEMBL29856915 0.90 KIT (0.61) BRAFKITBTKRAB9ANPC1
SCHEMBL29856172 0.87 BRAF (0.66) BRAFKITBTKRAB9ANPC1
SCHEMBL25245565 0.87 LMNA (0.56) BRAFKITMAPTLMNAABL1
SCHEMBL6184307 0.85 BRAF (0.82) BRAFKITABL1EGFRRET
SCHEMBL29562470 0.85 BRAF (0.82) BRAFKITABL1EGFRRET
SCHEMBL25802440 0.83 GAA (0.57) BRAFKITMAPTLMNAABL1
SCHEMBL30486132 0.83 LMNA (0.55) BRAFKITMAPTLMNAABL1
SCHEMBL16755338 0.80 KIT (0.78) BRAFKITABL1FGFR1KDR
SCHEMBL29856255 0.80 KIT (0.78) BRAFKITABL1FGFR1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111484482-B Alkynyl pyrimidine or alkynyl pyridine compound, and composition and application thereof 北京赛特明强医药科技有限公司 2022-06-21 CN disclosed