SCHEMBL29856468

SCHEMBL29856468

CCc1cc2ccnc(OC)c2n1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACSS2 Q9NR19 1/20 0.38
MAPT P10636 1/20 0.36
DYRK1A Q13627 4/20 0.32
MAOA P21397 1/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
RPS6KA5 O75582 1/20 0.32
TRPA1 O75762 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
DHFR P00374 1/20 0.31
HASPIN Q8TF76 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CCR1 P32246 1/20 0.30
CCR5 P51681 1/20 0.30
CCR8 P51685 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22502923 0.79 DYRK1A (0.37) MAPTDYRK1AMAOABCHEACHE
SCHEMBL24896258 0.73 KDM4E (0.50) ACSS2MAPT
SCHEMBL30220608 0.72 L3MBTL1 (0.50) MAPTMEN1KMT2A
SCHEMBL30593081 0.68 MAPT (0.40) ACSS2MAPTTRPA1CYP1A2CYP3A4
SCHEMBL22863378 0.68 MAPT (0.40) ACSS2MAPTTRPA1CYP1A2CYP3A4
SCHEMBL7016987 0.68 TLR8 (0.49) MAPTACHERPS6KA5TRPA1CYP1A2
SCHEMBL29856250 0.67 LOXL2 (0.39) MAPTDYRK1ATRPA1CYP1A2CYP3A4
SCHEMBL22502897 0.65 ALKBH5 (0.38) CYP1A2DHFRMEN1KMT2A
SCHEMBL21117365 0.65 CCR1 (0.31) CCR1CCR5CCR8
SCHEMBL9883177 0.65 ROCK1 (0.42) MAPTACHETRPA1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022169974-A1 INHIBITORS OF URAT1 AND PHARMACEUTICAL USES THEREOF NEXYS THERAPEUTICS, INC. (US) 2022-08-11 WO disclosed