SCHEMBL29856971

SCHEMBL29856971

COc1cc(=O)[nH]cc1C(=O)N(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.37
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 3/20 0.36
HPGD P15428 2/20 0.36
PDE9A O76083 1/20 0.36
CYP3A4 P08684 2/20 0.36
PAX8 Q06710 1/20 0.36
MAP4K1 Q92918 1/20 0.35
PDE3B Q13370 2/20 0.35
PDE3A Q14432 2/20 0.35
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35
PDE1C Q14123 1/20 0.35
PDE5A O76074 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
LRRK2 Q5S007 1/20 0.35
MAPK1 P28482 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20606051 0.81 ALDH1A1 (0.49) CHEK1ALDH1A1KDM4EHPGDCYP3A4
SCHEMBL28822756 0.79 KDM4E (0.41) CHEK1ALDH1A1KDM4EHPGDCYP3A4
SCHEMBL29856927 0.76 ALDH1A1 (0.34) ALDH1A1HPGDCYP3A4MAP4K1KEAP1
SCHEMBL14376019 0.74 CYP3A4 (0.57) ALDH1A1KDM4ECYP3A4PAX8PDE3B
SCHEMBL29465035 0.71 JAK2 (0.35) ALDH1A1PDE9ARECQLKEAP1
SCHEMBL22032380 0.71 SMN1; SMN2 (0.58) ALDH1A1KDM4EHPGDMAPK1KEAP1
SCHEMBL9793706 0.70 KDM4E (0.49) ALDH1A1KDM4ECYP3A4PAX8MAP4K1
Hydrochloric Acid SCHEMBL28822255 0.70 SMN1; SMN2 (0.57) ALDH1A1KDM4EHPGDMAPK1KEAP1
SCHEMBL1004370 0.69 PLAU (0.57) ALDH1A1KDM4EHPGDCYP3A4MAPT
SCHEMBL11653015 0.69 NPC1 (0.60) ALDH1A1HPGDCYP3A4PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109790146-B Pharmaceutical compounds 阿尔麦克探索有限公司 2022-08-23 CN disclosed