SCHEMBL28822756

SCHEMBL28822756

COc1cc(=O)[nH]cc1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 4/20 0.41
HPGD P15428 2/20 0.41
GAA P10253 2/20 0.41
GLA P06280 1/20 0.41
CHEK1 O14757 1/20 0.40
MAP2K2 P36507 1/20 0.40
MAP2K1 Q02750 1/20 0.40
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
CYP3A4 P08684 1/20 0.38
PARP15 Q460N3 2/20 0.37
PARP10 Q53GL7 2/20 0.37
TSHR P16473 1/20 0.37
APOBEC3A P31941 1/20 0.37
HTT P42858 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
NNMT P40261 1/20 0.37
POLB P06746 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20606051 0.84 ALDH1A1 (0.49) KDM4EALDH1A1HPGDGAACHEK1
SCHEMBL29856971 0.79 CHEK1 (0.37) KDM4EALDH1A1HPGDCHEK1CYP3A4
SCHEMBL26240985 0.76 MAP2K2 (0.42) KDM4EALDH1A1MAP2K2MAP2K1MKNK1
SCHEMBL12515332 0.74 CYP3A4 (0.52) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL28285146 0.72 CYP3A4 (0.61) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL30859597 0.71 KDM4E (0.47) KDM4EALDH1A1GAAGLAHTT
SCHEMBL6069006 0.69 LCK (0.60) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL9793655 0.69 KDM4E (0.53) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL33525781 0.69 ADRA1A (0.50) KDM4EALDH1A1GAACYP3A4TSHR
SCHEMBL6181459 0.68 KDM4E (0.51) KDM4EALDH1A1HPGDPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109195965-B Inhibitors of WDR5 protein-protein binding 普罗佩纶治疗公司 2022-07-26 CN disclosed